CAS: 96182-53-5; Tebupirimfos

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  • 51162-51-7 + 85929-96-0 = 96182-53-5
    反应条件:1.1 Reagents: Sodium Hydroxide Solvents: Toluene1.2 Catalysts: Benzyltributylammonium Chloride1.3 Reagents: Water
    标题:Process For The Production Of Dialkyl Pyrimidylphosphates
    参考文献:Canada]

    51162-51-7 + 85929-96-0 = 96182-53-5 [标题:Reaction Conditions
    标题:Phosphoric Acid Ester
    参考文献:Federal Republic Of Germany
📜2-叔丁基嘧啶-5-醇,Thiophosphorochloridic Acid O-Ethyl Ester O'-Isopropyl Ester 反应生成 丁基嘧啶磷
参考文献:Maurer,F.;Homeyer,B.;Becker,B.
标题:Maurer,F.;Homeyer,B.;Becker,B.

海关参考信息

专利信息


专利号:WO-2025056767-A1
优先权日:2023-09-15
标题 :Process for the preparation of enantiomerically enriched aliphatic amines
发明人:BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS
权利人:SYNGENTA CROP PROTECTION AG
摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.

专利号:US-2007232495-A1
优先权日:2006-03-24
标题:Compositions and methods to add value to plant products, increasing the commercial quality, resistance to external factors and polyphenol content thereof
发明人:NAPPA ALVARO O; LORENZINI FELIPE C; SANHUEZA ANDRES L
权利人:NAPPA ALVARO O; LORENZINI FELIPE C; SANHUEZA ANDRES L
摘要:The invention is related to compositions and methods that naturally protect plant tissues against ultraviolet radiation and temperature, thus giving protection against sunburn to plants, plant parts, fruits and/or flowers during their development. The invention is also related to compositions and methods to naturally improve the color of plants, plant parts, fruits and/or flowers by inducing the natural synthesis of flavonoids and anthocyanins present in plants. Likewise, the present invention is directed to improving the nutritional value of plants, plant parts, fruits and/or flowers by increasing the normal levels of polyphenolic compounds, especially flavonoids, present therein. Additionally, the present invention is related to compositions and methods that give more resistance to plants, plant parts, fruits and/or flowers against pathogens as bacteria and fungi. Finally, the present invention is related to plants, plant parts, fruits, flowers and/or propagating material treated with the compositions described in the present document.

专利号:WO-2021074309-A1
优先权日:2019-10-16
标 题:1-(3-quinolyl)-3,4-dihydroisoquinoline derivatives as fungicides for combating specific phytopathogens
发明人:WEISS MATTHIAS; QUARANTA LAURA; BOU HAMDAN FARHAN; MAHAJAN ATUL; WILLIAMS SIMON; KILARU JAGADEESH; SEN INDIRA; BIERI STEPHANE; DIGGELMANN MARTIN
权利人:SYNGENTA CROP PROTECTION AG
摘要:1-(3-quinolyl)-3,4-dihydroisoquinoline derivatives of formula (I) as well as a method of combating, preventing or controlling the phytopathogens Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale), which comprises applying to the phytopathogen, to the locus of the phytopathogen, or to a plant susceptible to attack by the phytopathogen, or to propagation material thereof, a fungicidally effective amount of a 1-(3-quinolyl)-3,4-dihydroisoquinoline derivative of formula (I). The present description discloses the synthesis of exemplary compounds, formulation examples, relevant biological data (antifungal activity against Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale) when spayed on plants), as well as comparative data against three prior art compounds (e.g. pages 52 to 85; formulation examples; examples A1 to A3; table E; compounds E.01 to E.187; biological examples). Exemplary compounds are e.g.: 5-bromo-1-(8-fluoro-3-quinolyl)spiro[4H-isoquinoline-3,1'- cyclopropane] (example A1) 5-bromo-1-(8-fluoro-3-quinolyl)-3,3-dimethyl-4H-isoquinoline (example A2) 1-(8-fluoro-3-quinolyl)-3,3-dimethyl-4H-isoquinoline-5-carbonitrile (example A3)

专利号:WO-2021074311-A1
优先权日:2019-10-16
标题:1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives as fungicides for combating specific phytopathogens
发明人:WEISS MATTHIAS; QUARANTA LAURA; BOU HAMDAN FARHAN; MAHAJAN ATUL; WILLIAMS SIMON; KILARU JAGADEESH; BIERI STEPHANE; DIGGELMANN MARTIN
权利人:SYNGENTA CROP PROTECTION AG
摘要:1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives of formula (I) as well as a method of combating, preventing or controlling the phytopathogens Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale), which comprises applying to the phytopathogen, to the locus of the phytopathogen, or to a plant susceptible to attack by the phytopathogen, or to propagation material thereof, a fungicidally effective amount of a 1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives of formula (I). The present description discloses the synthesis of exemplary compounds, formulation examples, relevant biological data (antifungal activity against Mycosphaerella graminicola, Monographella nivalis, Fusarium culmorum and/or Gibberella zeae when spayed on plants) (e.g. pages 47 to 55; examples A1 and A2; compounds E.01 to E.17; table E). An exemplary compounds is e.g.: 3-(5-bromo-3,3-dimethyl-2,4-dihydro-1 H-isoquinolin-1-yl)-8-fluoro- quinoline (example A1)

专利号:US-11213031-B2
优先权日:2017-11-13
标 题:Tetrazolylpropyl derivatives and their use as fungicides
发明人:SUDAU ALEXANDER; HOFFMANN SEBASTIAN; DAHMEN PETER; WEBSTER ROBERT ALAN; MEISSNER RUTH; GOERTZ ANDREAS; MILLER RICARDA; COQUERON PIERRE-YVES; BERNIER DAVID; NICOLAS LIONEL; BRUNET STEPHANE; KENNEL PHILIPPE; TOQUIN VALERIE; GOURGUES MATHIEU; LOQUE DOMINIQUE; THOMAS VINCENT
权利人:BAYER AG; BAYER CROPSCIENCE AG
摘要:The present invention relates to tetrazolylpropyl derivatives of formula (I) n nwherein one of V 1 and V 2 represents CR 3 and the other one of V 1 and V 2 represents N, Q represents a 6-membered aromatic cycle as defined in the specification, and R 1 , R 2 , R 3 , R 4 , and R 5 are defined as disclosed in the specification, to compositions comprising such compounds, to the use of said compounds as fungicides, as well as to particular intermediates useful in the synthesis of said tetrazolylpropyl derivatives.

专利号:BR-112019014061-A2
优先权日:2017-01-23
标 题 :compounds of formula i, intermediates b, intermediates c, intermediates ii and intermediates d, composition, use, method to combat phytopathogenic fungi, seed and process for the synthesis of the compounds of formula i

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主要参考文献


1: Use of High-throughput Enzyme-based Assay with Xenobiotic Metabolic Capability to Evaluate the Inhibition of Acetylcholinesterase Activity by Organophosphorus Pesticides Shuaizhang Li, Jinghua Zhao, Ruili Huang, Michael F. Santillo, Keith A. Houck, Menghang Xia Toxicol In Vitro. Author manuscript; available in PMC 2020 Apr 1.Published in final edited form as: Toxicol In Vitro. 2019 Apr;
56: 93–100. Published online 2019 Jan 6. doi: 10.1016/j.tiv.2019.01.002 Baumert, Megan Ulmer Carnes, Jane A. Hoppin, Chandra L. Jackson, Dale P. Sandler, Laura Beane Freeman, Paul K. Henneberger, David M. Umbach, Srishti Shrestha, Stuart Long, Stephanie J. London Sleep Health. Author manuscript; available in PMC 2019 Feb 1.Published in final edited form as: Sleep Health. 2018 Feb; 4(1): 20–26. Published online 2017 Sep 28. doi: 10.1016/j.sleh.2017.08.006 Hoppin, Stuart Long, David M. Umbach, Jay H. Lubin, Sarah Starks, Fred Gerr, Kent Thomas, Cynthia J Hines, Scott Weichenthal, Freya Kamel, Stella Koutros, Michael Alavanja, Laura E. Beane Freeman, Dale P. Sandler J Expo Sci Environ Epidemiol. Author manuscript; available in PMC 2013 May 1.Published in final edited form as: J Expo Sci Environ Epidemiol. 2012 Nov; 22(6): 584–592. Published online 2012 Aug 1. doi: 10.1038/jes.2012.79 Author manuscript; available in PMC 2013 Mar 18.Published in final edited form as: Neurotoxicol Teratol. 2012 Jan-Feb; 34(1): 168–176. Published online 2011 Aug 28. doi: 10.1016/j.ntt.2011.08.014 Hoppin, David M. Umbach, Stuart Long, Stephanie J. London, Paul K. Henneberger, Aaron Blair, Michael Alavanja, Laura E. Beane Freeman, Dale P. Sandler Environ Health Perspect. 2017 Apr; 125(4): 535–543. Published online 2016 Jul 6. doi: 10.1289/EHP315 Starks, Jane A. Hoppin, Freya Kamel, Charles F. Lynch, Michael P. Jones, Michael C. Alavanja, Dale P. Sandler, Fred Gerr Environ Health Perspect. 2012 Apr; 120(4): 515–520. Published online 2012 Jan 19. doi: 10.1289/ehp.1103944 Pardo, Laura E. Beane Freeman, Catherine C. Lerro, Gabriella Andreotti, Jonathan N. Hofmann, Christine G. Parks, Dale P. Sandler, Jay H. Lubin, Aaron Blair, Stella Koutros Environ Health. 2020;
19: 30. Published online 2020 Mar 5. doi: 10.1186/s12940-020-00583-0 2020;

合成参考文献


摘要:U.S. Environmental Protection Agency/Office of Prevention, Pesticides, and Toxic Substances. Reigart, J.R., Roberts, J.R. Recognition and Management of Pesticide Poisonings. 5th ed. 1999. EPA Document No. EPA 735-R-98-003, and available in electronic format at:
摘要:40 CFR 180.483; U.S. National Archives and Records Administration's Electronic Code of Federal Regulations. Available from, as of July 1, 2003:
摘要:Farm Chemicals Handbook 2001. Willoughby, Ohio: Meister 2001., p. C 380
摘要:IPCS; Poisons Information Monograph G001: Organophosphorus pesticides. (Date of last update: March 1998). Available from:
摘要:U.S. Environmental Protection Agency/Office of Prevention, Pesticides, and Toxic Substances. Reigart, J.R., Roberts, J.R. Recognition and Management of Pesticide Poisonings. 5th ed. 1999. EPA Document No. EPA 735-R-98-003, and available in electronic format at: https://www.epa.gov/pesticides/safety/healthcare, p. 40
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