CAS: 60607-34-3; 1-(3-(4-Benzhydrylpiperazin-1-yl)Propyl)-1,3-Dihydro-2H-Benzo[d]Imidazol-2-One

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CAS号841-77-0 二苯甲基哌嗪 | CAS号62780-89-6 1-(3-氯丙基)-1,3-二... | CAS号62781-00-4 N-(3-chloroprop... | CAS号100460-82-0 ethyl N-(3-chlo... | CAS号100460-83-1 N-ethoxycarbony... | CAS号100460-86-4 N-ethoxycarbony... | CAS号52099-72-6 1-异丙烯基-2-苯并咪唑酮 | CAS号102552-76-1 1-benzhydryl-4-... | CAS号776-74-9 二苯溴代甲烷 | CAS号100460-85-3 ethyl (2-aminop...

N-(3-氯丙基)-N-(2-硝基苯基)氨基甲酸乙酯置于palladium On Activated Charcoal Rac-4-Methyl-5-Methylhexan-2-One,氢气,Potassium Carbonate,Potassium Iodide,Calcium Chloride体系中,用 甲醇 作为反应溶剂,化学反应 5.5H,反应生成 奥沙米特
参考文献:Eine Neue Synthese Von 1-Alkyl-1,3-Dihydro-2H-Benzimidazol-2-Onen
标题:Eine Neue Synthese Von 1-Alkyl-1,3-Dihydro-2H-Benzimidazol-2-Onen
摘要:
DOI:10.1007/bf00798789

专利信息

专利号:US-6603003-B2
优先权日:2000-11-07
标 题 :Method for the preparation of piperazine and its derivatives
发明人：SEBASTIAN SONNY; PATEL HETAL VIRENDRA; THENNATI RAJAMANNAR
权利人:SUN PHARMACEUTICAL IND LTD
摘要:A novel method for the synthesis of piperazine and its derivatives of formula 1,wherein R is selected from hydrogen, or a lower alkyl group having 1 to 6 carbon atoms or a phenylalkyl group the alkyl of which has 1 to 4 carbon atoms;R1 is selected from hydrogen, a methyl group, a phenyl group optionally substituted with an alkyl group having 1 to 6 carbon atoms, or a phenylalkyl group the alkyl of which has 1 to 4 carbon atoms; andR2 is selected from hydrogen, or a methyl group, or a fluoromethyl group;comprising the steps:a. reacting an ester of formula 11 with substituted or unsubstituted ethylenediamine of formula 7 to give 3,4-dehydropiperazine-2-one and its derivatives of formula 12, wherein R, R1, R2 are as defined above and R6 is a C1 to C4 linear or branched alkyl group; andb. reacting the 3,4-dehydro-piperazine-2-one and its derivatives of formula 12 with a reducing agent to yield the piperazine and its derivatives of formula 1.

专利号:US-4678784-A
优先权日:1984-04-11
标题 :Method for the treatment of LHRH diseases and conditions
发明人：HO CHIH Y
权利人:MCNEILAB INC
摘要:Fused tetracyclic benzodiazepines of the formula (I): (I) where R1 is a cyclic amine such as 1-piperazine and R2 is H or a substituent as defined herein are useful as LHRH antagonizing agents. Also, methods for their synthesis, intermediates used in such synthesis, methods for use as medicaments and pharmaceutical compositions are described.

专利号:US-2023271983-A1
优先权日:2020-07-29
标题 :Functionalized isonitriles and products, preparation and uses thereof
发明人：SOTELO PÉREZ EDDY; AZUAJE GUERRERO JHONNY ALBERTO; MAJELLARO MARIA
权利人:UNIV SANTIAGO COMPOSTELA
摘要:The present invention relates to functionalized isonitrile compounds, formed by means of multicomponent environmentally friendly reactions, suitable for coupling to functional molecules such as biomolecules, APIs, chromophore and fluorophore molecules. The invention also relates to conjugates between said isonitrile compounds and functional molecules, which are useful in the synthesis of pharmaceutic drugs or tools, fluorescent molecules and labels, polymeric smart materials. The invention furthermore provides a kit for the in-vitro preparation of the functionalized isontrile compounds and conjugates. The invention also contemplates the medical use of said compounds and conjugates.

专利号:CN-104496739-A
优先权日:2014-11-24
标题 :Green Catalytic Synthesis of Diphenylmethane

专利号:US-4547497-A
优先权日:1984-04-11
标 题:Amidine benzodiazepines, methods for their use and intermediates
发明人：HO CHIH Y
权利人:MCNEILAB INC
摘要:Fused tetracyclic benzodiazepines of the formula (I): ##STR1## where R 1 is an acyclic amine or cyclic amine such as 1-piperidine, 4-morpholine or 1-piperazine and R 2 is H or a substituent as defined herein as useful as antiallergins. Also, methods for their synthesis, intermediate used in such synthesis, methods for use as medicaments and pharmaceutical compositions.

专利号:US-4587244-A
优先权日:1984-04-11
标 题 :Amidine benzodiazepines, methods for their use and intermediates
发明人：HO CHIH Y
权利人:MCNEILAB INC
摘要:Fused tetracyclic benzodiazepines of the formula (I): ##STR1## where R 1 is a cyclic amine such as 1-piperazine and R 2 is H or a substituent as defined herein are useful as antiovulatory and contragestational agents. Also, methods for their synthesis, intermediates used in such synthesis, methods for use as medicaments and pharmaceutical compositions are described.