CAS: 197855-65-5; Benzyl ((2S)-1-((4-Fluoro-3-Oxobutan-2-yl)Amino)-1-Oxo-3-Phenylpropan-2-yl)Carbamate

主要参考文献

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合成参考文献

参考文献:10.1124/mol.119.115964
摘要:Lee TD, Lee OW, Brimacombe KR, Chen L, Guha R, Lusvarghi S, Tebase BG, Klumpp-Thomas C, Robey RW, Ambudkar SV, Shen M, Gottesman MM, Hall MD. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. Molecular Pharmacology. 2019 Nov;96(5):629–40. doi: 10.1124/mol.119.115964.
参考文献:10.1021/jm00038a012
摘要:Wagner BM, Smith RA, Coles PJ, Copp LJ, Ernest MJ, Krantz A. In vivo inhibition of cathepsin B by peptidyl (acyloxy)methyl ketones. J Med Chem. 1994 Jun 10;37(12):1833–40. doi: 10.1021/jm00038a012.