CAS: 19005-93-7; 1H-Indole-2-Carbaldehyde

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CAS号24621-70-3 1H-吲哚-2-甲醇 | CAS号3770-50-1 吲哚-2-羧酸乙酯 | CAS号1477-50-5 吲哚-2-羧酸 | CAS号1202-04-6 吲哚-2-甲酸甲酯 | CAS号156571-69-6 N-甲氧基-N-甲基-1H-吲... | CAS号58881-45-1 1H-吲哚-2-羰酰氯 | CAS号1466-88-2 邻硝基肉桂醛 | CAS号144393-28-2 1-methoxymethox... | CAS号58881-41-7 Pyrazino[1,2-a;... | CAS号174418-78-1 1,2,3,4-tetrahy... | CAS号14255-18-6 1H-Indole,2-(2-... | CAS号146384-54-5 1-[(4-Methylphe... | CAS号3770-50-1 吲哚-2-羧酸乙酯 | CAS号74214-62-3 β-咔啉-3-羧酸乙酯(β-CCE) | CAS号80360-23-2 1-(苯磺酰)-1H-吲哚-2-甲醛 | CAS号27421-51-8 1-甲基吲哚-2-甲醛 | CAS号21109-25-1 1-(1H-吲哚-2-基)甲胺 | CAS号36193-65-4 2-氰基-1H-吲哚 | CAS号1477-50-5 吲哚-2-羧酸 | CAS号135440-68-5 3-[1-(2-叔丁氧基-2-...

1-(甲氧基甲氧基)吲哚置于palladium On Activated Charcoal 正丁基锂,氢气体系中,用 甲醇 用作溶剂,25.0 °C,101.33 Kpa 条件下,反应 0.33H,反应生成1H-吲哚-2-甲醛
参考文献:A Regioselective Lithiation Of 1-Methoxymethoxyindole At The 2-Position And Its Application For The Synthesis Of 2-Substituted Indoles
标题:A Regioselective Lithiation Of 1-Methoxymethoxyindole At The 2-Position And Its Application For The Synthesis Of 2-Substituted Indoles
摘要:A Regioselective Lithiation Of 1-Methoxymethoxyindole At The 2-Position Was Achieved With N-Buli At 0-Degrees-C. Subsequent Treatment With Electrophiles Afforded 2-Substituted 1-Methoxymethoxyindoles,Which Were Readily Converted To 2-Substituted Indoles.
Doi:10.3987/com-92-6066

专利信息

专利号:US-11427596-B2
优先权日:2019-07-19
标 题:Metal-free solvent-free synthesis of fused-pyrido heterocycles and biomedical applications
发明人：CHELVAM VENKATESH; DUDHE PREMANSH; KRISHNAN MENA ASHA; SONAWANE AVINASH
权利人:INDIAN INSTITUTE OF TECH INDORE
摘要:Embodiments herein provide fused-pyrido heterocycles such as azaindoles, carboline derivatives, furo[b]pyridines or furo[b]pyridine-isatin hybrids of Formula I.Embodiments also relate to a process for a synthesis of variety of complex pyrido-heterocycles The pyrido-heterocycles can be used for treating cancer (cervix, kidney, lung, breast and epidermal skin) and multi-drug resistant tuberculosis. These heterocycles can also be used as anti-biofilm agents against pathogenic strains, which will minimize the risk of secondary infections.

专利号:US-2016031800-A1
优先权日:2013-03-14
标 题:Synthesis of chiral kynurenine compounds and intermediates
发明人：TRETYAKOV ALEXANDER; DROUET KEITH E; SANDERS WILLIAM
权利人:VISTAGEN THERAPEUTICS INC
摘要:Provided are methods for the synthesis of compounds including chiral kynurenine compounds, intermediates useful for the synthesis thereof, and related compounds. For example, methods are provided for the synthesis of L-4-chlorokynurenine.

专利号:US-11427530-B2
优先权日:2018-02-09
标 题 :Synthesis of 4-chlorokynurenines and intermediates
发明人：LEVIN DANIEL; LEEMING PETER; EISENREICH EMERICH; LIU XUEJUN KARL
权利人:VISTAGEN THERAPEUTICS INC
摘要:The invention relates to an overall enantio-specific synthesis of 4-chlorokynurenine compounds, in particular L-4-chlorokynurenine, with improved yields. Large-scale syntheses are disclosed. The invention also relates to novel intermediates in the synthesis of L-4-chlorokynurenine.

专利号:US-5523411-A
优先权日:1994-03-14
标题 :Synthesis of mitomycin and its analogs
发明人：JIMENEZ LESLIE; WANG ZHENG
权利人:UNIV RUTGERS
摘要:The present invention relates to the synthesis of mitomycin and analogs thereof that are useful as anticancer antibiotics. The invention further relates to analogs of mitomycin, which can be prepared according to the methods of synthesis provided. The synthetic method of the invention provides for reacting a derivitized indole with a dialkylvinylsulfonium salt to yield a tricyclic skeleton having the precursors of the fourth ring in one step, followed by an oxidation step or steps to close the fourth ring and prepare mitomycin or a related compound.

专利号:US-9969685-B2
优先权日:2016-09-28
标 题 :Enantioselective synthesis of pyrroloindole compounds
发明人：SCHMIDT MICHAEL ANTHONY
权利人:BRISTOL MYERS SQUIBB CO
摘要:Compounds according to formula (I) or (II), wherein R 1 , R 2 , and R 3 are as defined in the specification, are versatile intermediates for the synthesis of DNA minor groove binder-alkylators having a cyclopropapyrroloindole (CPI) or seco-CPI alkylating subunit.

专利号:US-6133409-A
优先权日:1996-12-19
标 题:Process for the solid phase synthesis of aldehyde, ketone, oxime, amine, hydroxamic acid and αβ-unsaturated carboxylic acid and aldehyde compounds
发明人：SALVINO JOSEPH M; MORTON GEORGE C; MASON HELEN J; LABAUDINIERE RICHARD F
权利人:AVENTIS PHARM PROD INC
摘要:This invention is directed to a process for the solid phase synthesis of aldehyde, ketone, oxime, amine, hydroxamic acid and alpha , beta -unsaturated carboxylic acid and aldehyde compounds and to polymeric hydroxylamine resin compounds useful therefor.