CAS: 957061-16-4; 2-N,N-Diethylsulfamoylphenylboronic Acid
该化合物是一种多用途的碳酸衍生物,通常用于铃木-米亚乌拉交错反应,这是合成有机化学的一种关键方法,其独特的结构,在与博乐酸组相对的正方形位置上有一个二乙基硫磺基替代体,加强了酸组体的再活性和选择性.该化合物对于建立在制药,农用化学和材料科学中盛行的双亚基和异丙酸框架特别有用.电排的硫磺基组也可能影响试剂的稳定性和溶性,便于处理和净化.其定义明确的再活性特征使它成为复杂的分子合成的可靠建筑块.
- 英文名称2-N,N-Diethylsulfamoylphenylboronic Acid
- 中文名称[2-(二乙基氨磺酰基)苯基]硼酸
- IUPAC名称(2-(N,N-diethylsulfamoyl)phenyl)boronic acid
- 其它别名2-(N,N-二乙基氨磺酰)苯基硼酸; N,N-Diethyl 2-Boronobenzenesulfonamide
- CAS编号957061-16-4
- MFCD编号:MFCD09258634
- 分子式:C10H16BNO4S分子量:257.12
- 产品CID: 2011114
- 产品分类有机原料→分子砌块→芳环类化合物→苯类化合物
物理性质
MSDS等安全信息
合成工艺路线路线简述
海关参考信息
- 2902200000-苯
2901100000-饱和无环烃
2921199090-其他无环单胺 - 💡 提示：海关信息按照顺序优先匹配，如需确认的海关信息，请参考相关资料。
- 详情请参考：📖 海关编码查询和海关进出口税则
专利信息
专利号:US-9951062-B2
优先权日:2012-12-14
标 题 :Substituted 1 H-pyrrolo [2, 3-b] pyridine and 1 H-pyrazolo [3, 4-b] pyridine derivatives as salt inducible kinase 2 (SIK2) inhibitors
发明人：VANKAYALAPATI HARIPRASAD; YERRAMREDDY VENKATAKRISHNAREDDY; GANIPISETTY VENU BABU; TALLURI SURESHKUMAR; APPALANENI RAJENDRA P
权利人:ARRIEN PHARMACEUTICALS LLC
摘要:Compounds according to Formulas I, IA or IB: n nto pharmaceutically acceptable composition, salts thereof, their synthesis and their use as SIK2 inhibitors including such compounds and methods of using said compounds in the treatment of various diseases and/or disorders such as cancer, stroke, cardiovascular, obesity and type II diabetes.
