CAS: 170011-57-1; Tert-Butyl 4-(4-Aminophenyl)Piperidine-1-Carboxylate

相似化合物

454482-12-3 113310-52-4 387827-19-2

上下游产品

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4-氨基苯硼酸频哪醇酯置于palladium 10% On Activated Carbon,氢气,Sodium Carbonate体系中,用 甲醇,乙醇,水,甲苯 用作溶剂,80.0 °C,137.9 Kpa 条件下,反应 4.0H,反应生成1-Boc-4-(4-氨基苯基)哌啶
参考文献:Wo2020006075A5
标题:Wo2020006075A5

专利信息

专利号:WO-2025068371-A1
优先权日:2023-09-28
标 题:Inhibitors of the proprotein convertase furin, methods of production thereof and use
发明人：STEINMETZER TORSTEN; LANGE ROMAN WERNER; BOLLER CHARLOTTE; FRIEBERTSHÄUSER EVA; BLOCH KONSTANTIN
权利人:PHILIPPS UNIV MARBURG
摘要:The invention relates to novel inhibitors of the serine protease furin and to related furin-like proprotein convertases according to claim 1, and to methods of synthesis thereof and to use for production of medicaments for treatment of furin-dependent viral and bacterial infection diseases, and other disorders involving furin, such as cystic fibrosis, cancer, osteoarthritis, hypertension, and neurodegenerative disorders.