📜L-缬氨醇,4-(6-Chloroimidazo[1,2-B]Pyridazin-3-yl)Benzonitrile 以 N-甲基吡咯烷酮 作为反应溶剂,化学反应 0.5H,反应生成 琼脂糖凝胶cl-4B
参考文献:Synthesis And In Vitro Evaluation Of Imidazopyridazines As Novel Inhibitors Of The Malarial Kinase Pfpk7
标题:Synthesis And In Vitro Evaluation Of Imidazopyridazines As Novel Inhibitors Of The Malarial Kinase Pfpk7
摘要:A High-Throughput Screening Campaign Identified A Number Of Imidazopyridazines As Novel Inhibitors Of The Malarial Kinase Pfpk7. Further Synthetic Chemistry Efforts Enabled The Preparation Of A Number Of Analogues With Promising In Vitro Potencies. Although These Compounds Show Likely Broad Spectrum Inhibitory Activity,They Represent A Useful Starting Point For Further Chemical Optimisation. (C) 2008 Elsevier Ltd. All Rights Reserved.
DOI:10.1016/j.Bmcl.2008.08.043