专利号:US-9718764-B2 优先权日:2013-03-22 标题:Synthetic building blocks for the production of materials for organic electroluminescence devices 发明人:STOESSEL PHILIPP; PARHAM AMIR HOSSAIN; JATSCH ANJA 权利人:MERCK PATENT GMBH 摘要:The present invention relates to compounds which are suitable as synthesis precursors for the production of electronically active materials for use in organic electroluminescence devices.
专利号:US-2009137566-A1 优先权日:2005-05-26 标 题 :Substituted Piperdines as Renin Inhibitors 发明人:EHARA TAKERU; HITOMI YUKO; KONISHI KAZUHIDE; MASUYA KELICHI 权利人:EHARA TAKERU; HITOMI YUKO; KONISHI KAZUHIDE; MASUYA KELICHI 摘要:The invention relates to substituted 3,4- or higher substituted piperididine compounds, the use thereof for the preparation of a pharmaceutical formulation for the treatment of a disease that depends on activity of renin; the use of a compound of that class in the treatment of a disease that depends on activity of renin; these compounds for use in the diagnostic and therapeutic treatment of a warm-blooded animal, especially for the treatment of a disease (=disorder) that depends on activity of renin; pharmaceutical formulations or products comprising said compounds, and/or a method of treatment comprising administering said compounds, a method for the manufacture of said compounds, as well as novel intermediates, starting materials and/or partial steps for their synthesis. The compounds preferably have the formula I, n n n n n n n n n n wherein the moieties R1, R2, R11 and W are as defined in the specification.
专利号:US-10202374-B2 优先权日:2014-02-27 标题 :6-aryl-4-phenylamino-quinazoline analogs as phosphoinositide-3-kinase inhibitors 发明人:VISHWAKARMA RAM ASREY; BHARATE SANDIP BIBISHAN; BHUSHAN SHASHI; YADAV RAMMOHAN RAO; GURU SANTOSH KUMAR; JOSHI PRASHANT 权利人:COUNCIL SCIENT IND RES 摘要:The present invention relates to 6-aryl-4-phenylamino quinazolines of formula I wherein, R and R′ are as herein described. The present invention particularly relates to synthesis and anticancer and phoshpoinositide-3-kinase-α (PI3K-α) inhibitory activity. In addition, the invention relates to methods of using compounds for treating or preventing various cancers such as pancreatic, prostate, breast and melanoma.
专利号:CN-113788807-A 优先权日:2021-09-29 标 题:A kind of fused ring aromatic amine compound used in organic layer of OLED device and its synthesis method and application
摘要:Littke, A., Science of Synthesis: Cross Coupling and Heck-Type Reactions, (2012) 1, 258. 摘要:Lindh, J.; Larhed, M., Science of Synthesis: Cross Coupling and Heck-Type Reactions, (2012) 3, 280. 摘要:Xiao, X., Science of Synthesis: Knowledge Updates, (2023) 2, 199. 参考文献:10.1007/s10895-011-0896-1 摘要:Li XF, Chi ZG, Xu BJ, Li HY, Zhang XQ, Zhou W, Zhang Y, Liu SW, Xu JR. Synthesis and characterization of triphenylethylene derivatives with aggregation-induced emission characteristics. J Fluoresc. 2011 Sep;21(5):1969–77. doi: 10.1007/s10895-011-0896-1.