CAS: 16212-06-9; (E)-(2-(Phenylsulfonyl)Vinyl)Benzene

相似化合物

5418-11-1 129200-96-0 50709-88-1

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CAS号292638-84-7 phenylene-ethylene | CAS号873-55-2 苯亚磺酸钠 | CAS号515-42-4 苯磺酸钠 | CAS号536-74-3 苯乙炔 | CAS号591-50-4 碘苯 | CAS号5535-48-8 苯基乙烯基砜 | CAS号56069-39-7 苯砜基甲基膦酸二乙酯 | CAS号100-52-7 苯甲醛 | CAS号588-72-7 Benzene, [(1E)-... | CAS号2001-45-8 四苯基氯化膦 | CAS号673-32-5 1-苯基-1-丙炔 | CAS号5324-64-1 Benzene,[(2-phe... | CAS号3453-00-7 (2-氧代-2-苯乙基)膦酸二乙酯 | CAS号16212-05-8 烯丙基苯砜 | CAS号645-49-8 顺式-1,2二苯乙烯 | CAS号530-48-3 1,1-二苯基乙烯 | CAS号65885-18-9 [2-(benzenesulf... | CAS号65885-20-3 Benzenemethanam... | CAS号69333-48-8 [2-(benzenesulf...

📜(苯磺酰)乙酸置于苯甲醛体系中,用68%的收率获得反式苯基肉桂砜
参考文献:Styryl Sulfone Anticancer Agents
标题:Styryl Sulfone Anticancer Agents
摘要:本发明的苯乙烯基磺酰化合物选择性地抑制肿瘤细胞的增殖,并诱导肿瘤细胞凋亡,同时不损害正常细胞.这些化合物在治疗癌症和其他增殖性疾病中很有用,具有以下特征: (A) 公式ii: 其中n为零或一;R1选自氢,氯,氟和溴;R2选自氢,氯,氟,溴,甲基和甲氧基;R3选自氢,氯和氟;条件是,当r1和r3都是氢,N为零或一时,R2不能是甲基或甲氧基;且当n为一时,R1,R2和r3不能都是氢; (B) 公式iii: 其中r1选自氢,氯,氟和溴;或 (C) 公式iv: 其中r1选自氟和溴,R2选自2-氯苯基,4-氯苯基,4-氟苯基和2-硝基苯基.

专利信息

专利号:EP-2647639-A1
优先权日:2012-04-06
标题:ß-boration of alkene and alkyne intermediates
权利人:LEK PHARMACEUTICALS
摘要:The present invention relates to the field of organic chemistry, and in particular to the preparation of β-borated compounds. These β-borated compounds can be used as intermediates in the synthesis of pharmaceutically active agents such as Sitagliptin.

专利号:EP-2647640-A1
优先权日:2012-04-06
标 题:ß-boration of alkene and alkyne intermediates
权利人:LEK PHARMACEUTICALS
摘要:The present invention relates to the field of organic chemistry, and in particular to the preparation of β-borated compounds. These β-boated compounds can be used as intermediates in the synthesis of pharmaceutically active agents such as Sitagliptin.

专利号:US-5637719-A
优先权日:1989-06-09
标 题 :Reagents for rapid peptide synthesis
发明人：CARPINO LOUIS A; PHILBIN MICHAEL
权利人:RES CORP TECHNOLOGIES INC
摘要:The compounds of the present invention are adaptable as blocking or protecting groups for an amine composition useful in peptide synthesis. The present invention is directed to a method of protecting an amino group of an organic molecule during a reaction which modifies a portion of the molecule other than the protected amino group.

专利号:EP-0401817-B1
优先权日:1989-06-09
标题 :Reagents for rapid peptide synthesis
发明人：CARPINO LOUIS A; PHILBIN MICHAEL
权利人:RES CORP TECHNOLOGIES INC
摘要:This invention relates to compounds of the formula: wherein R is an electron withdrawing group; R1 is H or COZ; X1 and X2 are independently H, lower alkyl, aryl, aryl lower-alkyl or polystyrene or R and X1 taken together with the carbon atoms to which they are attached form a ring containing from 4 to 15 ring carbon atoms and may contain up to 2 heteroatoms, wherein the heteroatoms are O, S, or N; and Z is an amino acid residue, a peptide residue or a leaving group. The compounds of the present invention are adaptable as blocking or protecting groups for an amine composition useful in peptide synthesis. The present invention is also directed to a method of protecting an amino group of an organic molecule during a reaction which modifies a portion of the molecule other than the protected amino group.

专利号:KR-102325534-B1
优先权日:2019-10-11
标题 :Synthesis of Sulfones and Sulfonyl Derivatives using Sodium (tert-butyldimethylsilyl)oxymethanesulfinate

专利号:KR-20210043801-A
优先权日:2019-10-11
标 题 :Synthesis of Sulfones and Sulfonyl Derivatives using Sodium (tert-butyldimethylsilyl)oxymethanesulfinate