CAS: 64-95-9; 2-(Diethylamino)Ethyl 2,2-Diphenylacetate

上下游产品

2-Chloroethyl 2,2-Diphenylacetate 92907-17-0
二苯基乙酸甲酯 Methyl 2,2-Diphenylacetate 3469-00-9
2,2-二苯基乙酸 2,2-Diphenylacetic Acid 117-34-0

📜苯乙酸甲酯置于4-乙酰氨基苯磺酰叠氮,Sodium Carbonate,1,8-二氮杂双环[5.4.0]十一碳-7-烯,Potassium Hydroxide体系中,用 甲烷磺酸,二氯甲烷,1,2-二氯乙烷,乙腈 作为反应溶剂,化学反应 24.0H,反应生成 阿的芬宁
参考文献:蓝光辐照增强了芳基重氮乙酸酯与硼酸的室温偶联.
标题:蓝光辐照增强了芳基重氮乙酸酯与硼酸的室温偶联.
摘要:据报道可见光促进的光化学方案用于芳基重氮乙酸酯与硼酸的偶联.与没有光照的相同方案相比,这种光化学反应显示出极大的增强.除少数情况外,在黑暗(热过程)中的室温耦合通常不起作用.如果这样做的话,很可能还涉及到游离卡宾作为关键中间体.可替代地,光化学反应显示出广泛的范围,可以在空气中进行并且耐受各种各样的官能团.反应进化监测,Dft计算和控制实验已用于评估这种复杂机制的主要方面.具有生物活性的分子阿迪芬,苯那西嗪和阿普生已经被制备为合成应用的实例.
DOI:10.1002/chem.201905812

专利信息

专利号:US-2006030625-A1
优先权日:2004-08-06
标 题 :Dietary neurotransmitter precursors for balanced synthesis of neurotransmitters
发明人：HART CHERYLE RAM; GROSSMAN RONALD S; RAM HERBERT
权利人:HART CHERYLE RAM; GROSSMAN RONALD S; RAM HERBERT
摘要:Dietary supplements for treating a neurotransmitter deficiency include one or more precursors of the deficient neurotransmitter and a cofactor for activating in vivo enzymatic synthesis of the deficient neurotransmitter. The dietary supplements can also include an appropriate neurotransmitter, such as an amino acid. When administered through the oral mucosa, increases in levels of the deficient neurotransmitters and relief from deficiency symptoms are obtained.

专利号:US-6777554-B2
优先权日:2001-02-05
标题 :Preparation of N-methylparoxetine and related intermediate compounds
发明人：FINKELSTEIN NINA
权利人:TEVA PHARMA
摘要:The present invention provides a process for preparing N-methylparoxetine, an intermediate in the synthesis of paroxetine, by reacting sesamol-tetrabutylammonium salt with CIPMA. The present invention is not limited to the synthesis of N-methylparoxetine, but also includes other similar compounds.

专利号:WO-2009035652-A1
优先权日:2007-09-13
标 题 :Synthesis of deuterated catechols and benzo[d][1,3] dioxoles and derivatives thereof

专利号:US-7442386-B2
优先权日:2001-08-16
标题:Synthesis and use of reagents for improved DNA lipofection and/or slow release prodrug and drug therapies
发明人：DIAMOND SCOTT L; GRUNEICH JEFFREY ALAN
权利人:UNIV PENNSYLVANIA
摘要:The invention relates to compositions and methods for a one-step synthetic technique for making cationic steroid or cationic drug molecules for use as delivery vehicles. The invention further relates to methods for using cationic steroid molecules in lipofection or transfection, delivery of drugs, and for treatment of inflammation and other diseases and disorders. The invention also relates to cationic steroid prodrugs and cationic prodrugs and to methods of modifying drugs.

专利号:EP-2200997-A1
优先权日:2007-09-13
标 题:Synthesis of deuterated catechols and benzoýd¨ý1,3¨dioxoles and derivatives thereof

专利号:US-2009143432-A1
优先权日:2007-09-13
标 题:Synthesis of deuterated catechols and benzo[D][1,3]dioxoles and derivatives thereof