专利号:US-5514694-A 优先权日:1992-09-21 标题 :Peptidyl ketoamides 发明人:POWERS JAMES C; LI ZHAOZHAO; PATIL GIRISH S; CHU DER-LUN 权利人:GEORGIA TECH RES INST 摘要:A novel class of peptide alpha -ketoamides useful for selectively inhibiting serine proteases, selectively inhibiting cysteine proteases, generally inhibiting all serine proteases, and generally inhibiting all cysteine proteases, having the formula Y-CO-AA2-AA1-CO-NH-X. Processes for the synthesis of peptidyl alpha -ketoamide derivatives.
专利号:US-4141898-A 优先权日:1976-08-06 标题:Imidazo pyridinium quaternary salts as hypoglycemic agents 发明人:KUHLA DONALD E 权利人:PFIZER 摘要:The synthesis of imidazo[1,2-a]pyridinium, imidazo[1,5-a]pyridinium, pyrrolo[1,2-a]pyrazinium, pyrazolo[1,5-a]pyridinium, imidazo[2,1-a]isoquinolinium and imidazo[5,1-a]isoquinolinium quaternary salts and their use as hypoglycemic agents.
专利号:US-4044015-A 优先权日:1975-09-03 标题:Imidazopyridinium compounds as hypoglycemic agents 发明人:KUHLA DONALD E 权利人:PFIZER 摘要:The synthesis of imidazo[1,2-a]pyridinium, imidazo[1,5-a]pyridinium, pyrrolo[1,2-a]pyrazinium, pyrazolo[1,5-a]pyridinium, imidazo[2,1-a]isoquinolinium and imidazo[5,1-a]isoquinolinium quaternary salts and their use as hypoglycemic agents.
专利号:US-4163745-A 优先权日:1975-09-03 标 题:Imidazo[1,5-a]-quinolinium and imidazo[1,5-a]-pyridinium compounds 发明人:KUHLA DONALD E 权利人:PFIZER 摘要:The synthesis of imidazo[1,2-a]pyridinium, imidazo[1,5-a]pyridinium, pyrrolo[1,2-a]pyrazinium, pyrazolo[1,5-a]pyridinium, imidazo[2,1-a]isoquinolinium and imidazo[5,1-a]isoquinolinium quaternary salts and their use as hypoglycemic agents.
参考文献:10.1007/bf02242629 摘要:Mahmoud MM, Gray AR. Trypanosomiasis due toTrypanosoma evansi (steel, 1885) balbiani, 1888. a review of recent research. Tropical Animal Health and Production. 1980 Feb;12(1):35–47. doi: 10.1007/bf02242629.