📜二苯乙腈置于硫酸,Sodium Amide,苯体系中,化学反应生成 六氢-Alpha,Alpha-二苯基-1H-氮杂卓-1-丁酰胺 参考文献:Janssen Et Al.,Journal Of Medicinal And Pharmaceutical Chemistry,1959,Vol. 1,P. 187,189 标题:Janssen Et Al.,Journal Of Medicinal And Pharmaceutical Chemistry,1959,Vol. 1,P. 187,189
专利号:US-9982006-B2 优先权日:2014-08-21 标题:2′-chloro aminopyrimidinone and pyrimidine dione nucleosides 发明人:CLARKE MICHAEL O'NEIL HANRAHAN; MACKMAN RICHARD L; SIEGEL DUSTIN 权利人:GILEAD SCIENCES INC 摘要:Provided herein are formulations, methods and substituted 2′-chloro aminopyrimidinone and pyrimidine dione compounds of Formula (I) for treating Pneumovirinae virus infections, including respiratory syncytial virus infections, as well as methods and intermediates for synthesis of substituted 2′-chloro aminopyrimidinone and pyrimidine dione compounds.
专利号:US-9828388-B2 优先权日:2014-07-28 标题:Thieno[3,2-d]pyrimidine, furo[3,2-d]pyrimidine, and pyrrolo[3,2-D]pyrimidines useful for treating respiratory syncitial virus infections 发明人:CLARKE MICHAEL O'NEIL HANRAHAN; MACKMAN RICHARD L; SIEGEL DUSTIN 权利人:GILEAD SCIENCES INC 摘要:Provided herein are formulations, methods and substituted thieno[3,2-d]pyrimidine, furo[3,2-d]pyrimidine, and pyrrolo[3,2-d]pyrimidine compounds of Formula (I) for treating Pneumovirinae virus infections, including respiratory syncytial virus infections, as well as methods and intermediates for synthesis of substituted thieno[3,2-d]pyrimidine, furo[3,2-d]pyrimidine, and pyrrolo[3,2-d]pyrimidine compounds.
专利号:US-9701682-B2 优先权日:2013-11-11 标题:Pyrrolo[1,2-f][1,2,4]triazines useful for treating respiratory syncitial virus infections 发明人:CLARKE MICHAEL O'NEIL HANRAHAN; DOERFFLER EDWARD; MACKMAN RICHARD L; SIEGEL DUSTIN 权利人:GILEAD SCIENCES INC 摘要:Provided herein are formulations, methods and substituted tetrahydrofuranyl-pyrrolo[1,2-f][1,2,4]triazine-4-amine compounds of Formula (I) for treating Pneumovirinae virus infections, including respiratory syncytial virus infections, as well as methods and intermediates for synthesis of tetrahydrofuranyl-pyrrolo[1,2-f][1,2,4]triazine-4-amine compounds.
1. Kalanur SS, Seetharamappa J, Prashanth SN. Interaction of an antidepressant buzepide methiodide with DNA immobilized on the glassy carbon electrode. Colloids Surf B Biointerfaces. 2011 Feb 1;82(2):438-42. doi: 10.1016/j.colsurfb.2010.09.017. Epub 2010 Sep 29.