专利号:US-8962863-B2 优先权日:2012-08-21 标 题:Process for the synthesis of substituted gamma lactams 发明人:DINH DANNY T; GARST MICHAEL E; OLD DAVID W; SYAGE ELIZABETH T; GORIN BORIS; LANTHIER CHRISTOPHER M; OUDENES JAN 权利人:ALLERGAN INC 摘要:The present invention provides synthetic processes for the preparation of a variety of well-defined substituted gamma lactams. The compounds that can be prepared by the process of the invention are useful for treating a variety of conditions. In some embodiments of the invention, the compounds are useful for treating ocular disorders, such as, for example, glaucoma, lowering of elevated intraocular pressure, and the like. In other embodiments, the compounds are useful for treating irritable bowel disease. In further embodiments, the compounds are useful in promoting hair growth. In still further embodiments, the compounds are useful in promoting wound healing, scar reduction, and the like.
专利号:EP-3515880-B1 优先权日:2017-03-17 标题:Methods and compositions for synthesis of encoded libraries 发明人:LI JIN; MORGAN BARRY A; Wan jinqiao; DOU DENGFENG; LIU GUANSAI; CHANG YONG; CHEN QIUXIA; WANG XING; XU YANSHAN; HU DONGYAN; LIU JIAN; CHENG XUEMIN 权利人:HITGEN INC
专利号:US-2020149034-A1 优先权日:2017-03-17 标题:Methods and Compositions for Synthesis of Encoded Libraries
专利号:US-2014058117-A1 优先权日:2012-08-21 标 题 :Process for the synthesis of substituted gamma lactams
专利号:KR-102221534-B1 优先权日:2012-08-21 标题:Process for the synthesis of substituted gamma lactams
专利号:CA-3170288-A1 优先权日:2020-03-04 标题:Synthesis of novel ep4 antagonist and use in cancer and inflammation
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