CAS: 253-45-2; 2,7-Naphthyridine

相似化合物

86278-61-7 1309379-44-9 28002-16-6

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CAS号222167-81-9 4-(2-trimethyls... | CAS号1120-87-2 4-溴吡啶 | CAS号154105-64-3 4-溴吡啶-3-甲醛 | CAS号100135-62-4 3-Dicyanmethyle... | CAS号105-50-0 丙酮二羧酸二乙酯 | CAS号69042-30-4 1-氯-2,7-萘啶 | CAS号3222-50-2 4-甲基吡啶-3-羧酸 | CAS号67988-50-5 2,7-萘啶-1(2H)-酮 | CAS号6790-32-5 龙胆定碱 | CAS号853648-79-0 2,7-Naphthyridi... | CAS号108749-08-2 1,2,3,4-四氢-2,7-萘啶

📜4-溴吡啶置于bis-Triphenylphosphine-Palladium(II) Chloride,Copper(L) Iodide,氨,三乙胺,Lithium Diisopropyl Amide体系中,用 四氢呋喃,乙醇,N,N-二甲基甲酰胺 用作溶剂,化学反应 10.5H,反应生成2,7-萘啶
参考文献:二氮杂萘通过ch取代的一锅均和交叉偶联:双和三重氮杂萘的合成
标题:二氮杂萘通过ch取代的一锅均和交叉偶联:双和三重氮杂萘的合成
摘要:仅使用四甲基哌啶锂(litmp)试剂研究了未活化的重氮萘的无过渡金属偶联反应.对称和不对称的双二氮杂萘通过相关单体的均相和交叉偶联以中等至高收率合成.另外,使用适当当量的litmp进行了二喹喔啉[2,3-A:2',3'C]吩嗪和2,2':3',2''-Terquinoxaline的一步合成.通过NMR光谱和hrms光谱对产物进行表征.
Doi:10.1002/jhet.4111

专利信息

专利号:US-2006009510-A1
优先权日:2004-07-09
标 题 :Method of synthesizing indolinone compounds
发明人：HAVENS JEFFREY L; VAIDYANATHAN RAJAPPA
权利人:PHARMACIA & UPJOHN CO LLC
摘要:Disclosed are methods of preparing pyrrole compounds of formula 14 and indolinone compounds of formula 1 n nvia a synthetic route wherein the amide sidechain on the pyrrole moiety is attached prior to pyrrole formation. The compounds 14 produced by the methods herein are useful in the synthesis of compounds of formula 1, which are useful in the treatment of abnormal cell growth, such as cancer.

专利号:US-7763734-B2
优先权日:2006-04-19
标题 :Synthesis, structure and use of bisoxazolidines for asymmetric catalysis and synthesis
发明人：WOLF CHRISTIAN; LIU SHUANGLONG
权利人:UNIV GEORGETOWN
摘要:One aspect of the invention relates to chiral bisoxazolidines and their use in asymmetric catalysis. The chiral bisoxazolidines are a novel class of compounds that is expected to find multiple applications, for example, in asymmetric synthesis. For example, a bisoxazolidine ligand enabled the catalytic enantioselective alkynylation and alkylation of a range of aromatic and aliphatic aldehydes, generating chiral propargylic alcohols and secondary alcohols in high yields and enantiomeric excess.

专利号:US-11976052-B2
优先权日:2019-01-11
标题:Leukotriene synthesis inhibitors
发明人：BURGOYNE DAVID L; DEBRUIN ERIN; FONAREV JULIA; YEE JAMES GEE KEN; LANGLANDS JOHN MICHAEL
权利人:NAEGIS PHARMACEUTICALS INC
摘要:Provided are specific leukotriene synthesis inhibitor compounds and pharmaceutical compositions comprising the compounds and methods of using the compounds and the pharmaceutical compositions in treating, for example, inflammatory diseases or conditions.

专利号:US-10233182-B2
优先权日:2014-04-04
标题 :Substituted spirocyclic inhibitors of autotaxin
发明人：BABISS LEE; CLARK MATTHEW; KEEFE ANTHONY D; MULVIHILL MARK J; NI HAIHONG; RENZETTI LOUIS; RUEBSAM FRANK; WANG CE; XIE ZHIFENG; ZHANG YING
权利人:X RX INC
摘要:The present invention relates to compounds according to Formula I and pharmaceutically acceptable salts, synthesis, intermediates, formulations, and methods of disease treatment therewith, including cancer, lymphocyte homing, chronic inflammation, neuropathic pain, fibrotic diseases, thrombosis, and cholestatic pruritus, mediated at least in part by ATX.

专利号:US-2016326157-A1
优先权日:2014-01-06
标 题:Monobactams and methods of their synthesis and use
发明人：MYERS ANDREW G; Seiple lan Bass; SUSSMAN ROBIN JUDITH
权利人:HARVARD COLLEGE
摘要:Described herein are monobactam antibiotics of Formula (I), (I′), (II), and (II′), along with methods and intermediates for preparing these compounds. Pharmaceutical compositions and methods of treating infectious diseases using the monobactams are also provided.

专利号:US-4416817-A
优先权日:1979-06-08
标题:3-Methoxy-2-oxoazetidine derivatives and their production
发明人：MATSUO TAISUKE; OCHIAI MICHIHIKO
权利人:TAKEDA CHEMICAL INDUSTRIES LTD
摘要:Novel 3-methoxy-2-oxoazetidine derivatives, which are shown by the following formula wherein R1 is amino, acylated amino or protected amino, are of value as intermediates for the synthesis of useful compounds represented by the formula wherein R1 has the same meaning as defined above, as drugs in the treatment of bacterial infections.