专利号:WO-0140193-A1 优先权日:1999-12-03 标题:Method for the synthesis of pyrazolines 发明人:BOLDI ARMEN M 权利人:CHEMRX ADVANCED TECHNOLOGIES I; BOLDI ARMEN M 摘要:The present invention provides a method for the synthesis of compounds of Formula (I). Also claimed are novel intermediates and their methods of synthesis.
专利号:US-2002103381-A1 优先权日:2000-11-30 标 题 :Method for the synthesis of pyrazolines 发明人:BOLDI ARMEN M 摘要:The present invention provides a method for the synthesis of compounds of Formula I: n n n Also claimed are novel intermediates and their methods of synthesis.
专利号:US-5859288-A 优先权日:1995-03-24 标 题:Reagent and process for the synthesis of oxysulphide-containing fluorine-containing organic derivatives 发明人:FORAT GERARD; MAS JEAN-MANUEL; SAINT-JALMES LAURENT 权利人:RHONE POULENC CHIMIE 摘要:The invention relates to a reagent which is useful for the synthesis of oxysulphide-containing fluorine-containing organic derivatives by reacting with an oxide of sulphur, especially sulphur dioxide, characterized in that it comprises: a) a fluorocarboxylic acid of formula Ew-CF2-COOH where Ew is an electron-withdrawing group or atom which is at least partially salified by an organic or inorganic cation, and b) an aprotic polar solvent; and in that the content of releasable protons carried by its various components, including their impurities, is at most equal to half the initial molar concentration of the said fluorocarboxylic acid. This reagent can be used by heating in order to form fluorine-containing sulphinic or sulphonic acids.
专利号:WO-0056721-A1 优先权日:1999-03-23 标题 :Solid phase synthesis of benzodiazepine diones 发明人:DENER JEFFREY MARK 权利人:AXYS PHARM INC; DENER JEFFREY MARK 摘要:The present invention provides a process for the synthesis of a compound or an array of compounds of formula (I). Compounds of formula (I) generally represent the therapeutically important class of compounds namely diversely substituted benzodiazepine diones.
专利号:WO-0168615-A1 优先权日:2000-03-13 标题 :Quinazoline synthesis 发明人:DENER JEFFREY MARK; LEASE TIMOTHY G; NOVACK AARON ROBERT 权利人:CHEMRX ADVANCED TECHNOLOGIES I; DENER JEFFREY MARK; LEASE TIMOTHY G; NOVACK AARON ROBERT 摘要:The present invention relates to a method for making a compound of Formulas I, II and III. The method of the present invention also enables parallel and simultaneous synthesis of a plurality of compounds represented by Formulas I, II and III.
专利号:WO-2021148594-A1 优先权日:2020-01-23 标题 :Chemical synthesis of the peptidic part of bioactive natural products 发明人:RACINE EMILIE 权利人:NOSOPHARM 摘要:The present invention relates to a method for preparing a peptide of following general formula (I). It also relates to specific peptides, which have been prepared by the method according to the invention, and key synthesis intermediates.
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合成参考文献
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