CAS: 153624-46-5; 4-Isopropoxyphenylboronic Acid

相似化合物

176672-49-4 22237-13-4 216485-86-8

上下游产品

CAS号6967-88-0 4-异丙氧基溴苯 | CAS号121-43-7 硼酸三甲酯 | CAS号1044239-22-6 5-[4-(异丙氧基)苯基]-2-吡啶胺

1-溴-4-异丙氧基苯置于叔丁基锂,硼酸三甲酯体系中,用 四氢呋喃 用作溶剂,以71%的收率获得4-异丙氧基苯硼酸
参考文献:Palladium-Catalyzed Cross-Coupling Of N-Benzenesulfonyl-3,4-Dibromopyrrole And Its Application To The Total Syntheses Of Lamellarins O,P,Q,And R
标题:Palladium-Catalyzed Cross-Coupling Of N-Benzenesulfonyl-3,4-Dibromopyrrole And Its Application To The Total Syntheses Of Lamellarins O,P,Q,And R
摘要:Palladium-Catalyzed Suzuki-Miyaura Coupling Of N-Benzenesulfonyl-3,4-Dibromopyrrole With A Variety Of Arylboronic Acids Gave The Corresponding 3,4-Diarylpyrroles In High Yields. The 3,4-Differentially Arylated Pyrroles Could Also Be Prepared By Stepwise Cross-Coupling Approach. The Total Syntheses Of Lamellarins O,P,Q,And R Have Been Achieved By Using The Cross-Coupling And The Directed Lithiation As Key Reactions. (C) 2007 Elsevier Ltd. All Rights Reserved.
Doi:10.1016/j.Tet.2007.10.105

专利信息

专利号:US-2006287529-A1
优先权日:2003-02-20
标 题:Solid phase synthesis of antitumoral compounds
发明人：ALVAREZ MERCEDES; ALBERICIO FERNANDO; CIRONI PABLO; CUE VAS CARMEN; FRANCESCH ANDREAS; MARFIL MARTA
权利人:ALVAREZ MERCEDES; ALBERICIO FERNANDO; CIRONI PABLO; CUE VAS CARMEN; FRANCESCH ANDREAS; MARFIL MARTA
摘要:Lamellarins are prepared using a solid phase synthesis. In a first aspect, the process includes a step as follows: Formula (I) where R 1 to R 15 are as defined, and X is halogen, provided that one of R 2 , R 3 or R 4 is immobilised to a resin. In a second aspect, the process includes a step as follows: Formula (II) where R 1 ′ to R 5 ′, R 11 ′ and R 13 ′ are as defined, X 1 and X 2 are halogen, M is a metal function and PG is an amino protecting group, provided that one of that R 2 ′, R 3 ′ or R 4 ′ is immobilised to a resin.

专利号:US-9994550-B2
优先权日:2014-01-07
标题 :Heterocyclic modulators of lipid synthesis for use against cancer and viral infections
发明人：WAGMAN ALLAN S; JOHNSON RUSSELL J; ZAHARIA CRISTIANA A; CAI HAIYING; HU LILY W; DUKE GREG; OHOL-GUPTA YAMINI; HEUER TIMOTHY; O'FARRELL MARIE
权利人:3 V BIOSCIENCES INC
摘要:Heterocyclic modulators of lipid synthesis are provided as well as pharmaceutically acceptable salts thereof; pharmaceutical compositions comprising such compounds; and methods of treating conditions characterized by dysregulation of a fatty acid synthase pathway by the administration of such compounds.

专利号:EP-1613635-A2
优先权日:2003-02-20
标题 :Solid phase synthesis of antitumoral compounds

专利号:AU-2004212762-A1
优先权日:2003-02-20
标 题:Solid phase synthesis of antitumoral compounds

专利号:CA-2515313-A1
优先权日:2003-02-20
标 题 :Solid phase synthesis of antitumoral compounds

专利号:WO-2004073598-A2
优先权日:2003-02-20
标题 :Solid phase synthesis of antitumoral compounds