专利号:US-9446995-B2 优先权日:2012-05-21 标 题:Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions 发明人:CHONG HYUN-SOON 权利人:CHONG HYUN-SOON; ILLINOIS INST OF TECH 摘要:Stereoselective and regioselective synthesis of compounds via nucleophilic ring opening reactions of aziridinium ions for use in stereoselective and regioselective synthesis of therapeutic and diagnostic compounds.
专利号:US-10189803-B2 优先权日:2008-02-22 标题 :Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions 发明人:CHONG HYUN-SOON 权利人:CHONG HYUN SOON; ILLINOIS INSTITUTE OF TECH 摘要:Stereoselective and regioselective synthesis of compounds via nucleophilic ring opening reactions of aziridinium ions for use in stereoselective and regioselective synthesis of therapeutic and diagnostic compounds.
专利号:EP-3599246-A1 优先权日:2018-07-25 标题 :Means and methods for synthesizing precursors of y-aminobutyric acid (gaba) analogs 发明人:POELARENDS GERRIT JAN; BIEWENGA LIEUWE; VAN DER MEER JAN-YTZEN; PODDAR HARSHWARDHAN; THANGAVELU SARAVANAN 权利人:UNIV GRONINGEN 摘要:The invention relates to the fields of drug development and biocatalysis, more specifically to a biocatalytic route for asymmetric synthesis of precursors of y-aminobutyric acid (GABA) analogs. Provided is an isolated mutant 4-oxalocrototonate tautomerase (4-OT) enzyme comprising the following mutations (i) leucine at position 8 substituted with a tyrosine (L8Y) or a phenylalanine (L8F); (ii) methionine at position 45 substituted with a tyrosine (M45Y); and (iii) phenylalanine at position 50 substituted with an alanine (F50A), wherein the positions are numbered according to the amino acid sequence of 4-OT ofPseudomonas putida.Also provided is a method for the synthesis of a precursor for the pharmaceutically relevant enantiomer of a GABA analog, comprising (i) providing a y-nitroaldehyde using the 4-OT mutant enzyme, followed by (ii) subjecting the thus obtained y-nitroaldehyde to an enzymatic oxidation reaction catalyzed by an aldehyde dehydrogenase (EC 1.2.1.3).
专利号:US-2013310555-A1 优先权日:2012-05-21 标题:Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions
专利号:CN-120041848-A 优先权日:2025-02-18 标 题 :Method for electrochemically synthesizing chiral beta-ester nitrile and application of chiral beta-ester nitrile in synthesis of baclofen and rolipram
专利号:US-2017008863-A1 优先权日:2008-02-22 标 题:Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions
1: Nadarajan D, O'Brien J, Cresswell S, Kele B, Mueller J, Bade R. Application of design of experiment for quantification of 71 new psychoactive substances in influent wastewater. Anal Chim Acta. 2024 Sep 8;1321:343036. doi: 10.1016/j.aca.2024.343036. Epub 2024 Jul 30. 2024:8824770. doi: 10.1155/2024/8824770. 3: Long T, Gollamudi S, Pai S; ACCP Public Policy Committee. ACCP Position Statement on Unregulated Psychotropic Products. J Clin Pharmacol. 2024 Aug;64(8):905-907. doi: 10.1002/jcph.2485. Epub 2024 Jul 2. 19(11):e202400064. doi: 10.1002/asia.202400064. Epub 2024 May 6.
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