专利号:US-6521664-B1 优先权日:1999-12-08 标 题:Pesticidal activity of functionalized alkenes 发明人:LINDERMAN RUSSELL J 权利人:UNIV NORTH CAROLINA STATE 摘要:The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as “pesticidal compoundsâ€?). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
专利号:WO-2025056767-A1 优先权日:2023-09-15 标题 :Process for the preparation of enantiomerically enriched aliphatic amines 发明人:BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS 权利人:SYNGENTA CROP PROTECTION AG 摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.
专利号:EP-0590361-A1 优先权日:1992-09-17 标 题 :Process for the preparation of 2-amino-6-halopurines 发明人:HAGEN HELMUT DR; RAATZ PETER DR 权利人:BASF AG 摘要:Preparation of 2-amino-6-halopurines I (X = halogen) by hydrolysis of 2-acylamino-6-halopurines II (R¹, R² = acyl; R² = H) in the presence of an acid or base and preparation of II by acylation of guanine III to acylguanine Va or Vb and halogenation of V with a halogenating agent VI to II.n n n V and II are new intermediates for the synthesis of I when R1 and R2 are haloacetyl.
专利号:US-6660770-B2 优先权日:1999-12-08 标题:Pesticidal activity of functionalized alkenes 发明人:LINDERMAN RUSSELL J; ROE R MICHAEL; THOMPSON DEBORAH M; VANDERHEREHEN MATTHEW 权利人:UNIV NORTH CAROLINA STATE 摘要:The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as “pesticidal compoundsâ€?). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
专利号:US-10906880-B2 优先权日:2016-01-26 标题:Kind of isothiazole oxime ether-containing strobilurin derivatives and its preparation methods and application 发明人:FAN ZHIJIN; CHEN LAI; GUO XIAOFENG; ZHU YUJIE; QIAN XIAOLIN; MA LIUYONG; ZHANG NAILOU; WANG HAIXIA; ZHANG ZHIMING; XU JINGHUA; SONG YINQI 权利人:UNIV NANKAI 摘要:The present invention is that provided a synthesis method of a series of isothiazole oxime ether containing strobilurin derivatives IV. The present invention relates to 3,4-dichloroisothiazolyl oxime ether strobilurin derivatives, and their chemical structural formula is as shown by IV. n n n n n n n n n n The invention discloses the structural formula of the above compound, the synthesis method and the use as an insecticide, a fungicide, an anti-plant virus agent, and an agriculturally acceptable auxiliary or synergist and a commercial insecticide. The use of a fungicide, an anti-plant virus agent and an acaricide in combination for controlling agricultural, forestry, horticultural plant pests, diseases, virus diseases and preparation methods.
专利号:EA-023329-B1 优先权日:2012-12-06 标 题 :METHOD OF SYNTHESIS OF 3- (2-BROM-4,5-DIMETOXYPHENYL) PROPNANITRIL AND APPLICATION IN THE SYNTHESIS OF IVABRADIN AND ITS PHARMACEUTICAL ACCEPTABLE ACID ADDITIVE SALTS
1: Hoang TC, Rand GM. Mosquito control insecticides: a probabilistic ecological risk assessment on drift exposures of naled, dichlorvos (naled metabolite) and permethrin to adult butterflies. Sci Total Environ. 2015 Jan 1;502:252-65. doi: 10.1016/j.scitotenv.2014.09.027. Epub 2014 Sep 26. doi: 10.1016/j.chemosphere.2014.10.040. Epub 2014 Nov 11. doi: 10.1002/etc.1757. Epub 2012 Feb 24. doi: 10.1016/j.pestbp.2016.02.001. Epub 2016 Feb 4. doi: 10.1007/s00244-009-9353-4. Epub 2009 Jun 18. doi: 10.1007/s10646-010-0497-9. Epub 2010 Apr 29. doi: 10.1603/EN10089. doi: 10.1002/ieam.1534. Epub 2014 May 29. German. doi: 10.1603/EN09087. doi: 10.1007/s10646-014-1402-8. Epub 2014 Dec 20.
合成参考文献
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