专利号:US-8742118-B2 优先权日:2011-10-27 标题 :Methods for preparing intermediates of perampanel 发明人:FONTANA FRANCESCO; STABILE PAOLO 权利人:F I S —FABBRICA ITALIANA SINT S P A 摘要:Methods for the synthesis of 2-alkoxy-5-(pyridin-2-yl)pyridine of formula I n nor salts thereof are provided.
专利号:US-10111867-B2 优先权日:2015-02-17 标题:Process and intermediates for the preparation of perampanel 发明人:MAROM EHUD; RUBNOV SHAI 权利人:MAPI PHARMA LTD 摘要:The present invention describes a process for the synthesis of 3-(2-cyanophenyl)-5-(2-pyridyl)-1-phenyl-1,2-di-hydro-pyridin-2-one (Perampanel) represented by the structure of formula (1), and salts thereof, especially salts with pharmaceutically acceptable acids. The present invention further relates to certain intermediates formed and/or used in such process.
专利号:CN-109096181-B 优先权日:2018-09-29 标题:A method for ultrasonic-assisted green synthesis of 2-sulfonylpyridine derivatives
专利号:CN-114478368-A 优先权日:2022-01-21 标 题 :Synthesis method and application of a kind of chiral paramagnetic probe Py-D-Cys-DTPA
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