CAS: 63285-84-7; 3-Phenoxythiophene

上下游产品

3-Bromothiophene phenol 3-phenoxythiophene-2-carboxylic acid 4-phenoxythiophene-2-carboxylic acid 3-phenoxythiophene-2,5-dicarboxylic acid 3-phenoxythiophene-2-sulfonyl chloride

📜3-溴噻吩,苯酚置于氯化亚铜体系中,用 吡啶,Mineral Oil 作为反应溶剂,以74%的收率获得产物3-苯氧基噻吩
参考文献:Thienyl-,Furyl-And Pyrrolyl Sulfonamides And Derivatives Thereof That
标题:Thienyl-,Furyl-And Pyrrolyl Sulfonamides And Derivatives Thereof That
摘要:提供了噻吩基,呋喃基和吡咯基磺酰胺以及调节或改变内皮素家族肽活性的方法.具体来说,提供了n-(异噁唑基)噻吩磺酰胺,N-(异噁唑基)呋喃磺酰胺和n-(异噁唑基)吡咯磺酰胺,以及使用这些磺酰胺通过将其与受体接触来抑制内皮素肽与内皮素受体结合的方法.还提供了通过给予这些磺酰胺或其前药的有效量来治疗内皮素介导的疾病的方法,这些磺酰胺或其前药可以抑制或增加内皮素的活性.

专利信息

专利号:US-2008280855-A1
优先权日:2005-06-22
标 题 :Process For the Production of Intermediates For the Preparation of Tricyclic Benzimidazoles
发明人：CHIESA MARIA VITTORIA; PALMER ANDREAS; BUHR WILM; ZIMMERMANN PETER JAN; BREHM CHRISTOF; SIMON WOLFGANG-ALEXANDER; POSTIUS STEFAN; KROMER WOLFGANG; ZANOTTI-GEROSA ANTONIO
权利人:NYCOMED GMBH
摘要:The invention relates to a process for the synthesis of compounds of the formula 1-a and compounds of the formula 1-b. n n n n n n n n n n The compounds of the formula 1-a and the compounds of the formula 1-b, in which the substituents R1, R2, R3, and Ar have the meanings indicated in the description, are valuable intermediates for the preparation of pharmaceutically active compounds.

专利号:WO-2007141253-A1
优先权日:2006-06-07
标 题 :Process for the production of intermediates for the preparation of tricyclic imidazopyridines
发明人：PALMER ANDREAS; BUHR WILM; ZIMMERMANN PETER JAN; BREHM CHRISTOF; CHIESA MARIA VITTORIA; ZANOTTI-GEROSA ANTONIO
权利人:NYCOMED GMBH; PALMER ANDREAS; BUHR WILM; ZIMMERMANN PETER JAN; BREHM CHRISTOF; CHIESA MARIA VITTORIA; ZANOTTI-GEROSA ANTONIO
摘要:The invention relates to a process for the synthesis of compounds of the formula (1-a) and compounds of the formula (1-b). The compounds of the formula 1-a and the compounds of the formula 1-b, in which the substituents R1, R2, R3, and Arom have the meanings indicated in the description, are valuable intermediates for the preparation of pharmaceutically active compounds.

专利号:US-2008281105-A1
优先权日:2005-01-18
标题:Novel Quinolinium Salts and Derivatives
发明人：MACDONALD JAMES E; HYSELL MICHELLE K; YU DEHUA; LI HENRY; WONG-STAAL FLOSSIE
权利人:IMMUSOL INC
摘要:The present invention relates generally to the synthesis of novel quinolinium salts and derivative compounds. Such salts and compounds are useful for inhibiting the growth of cancer cells.

专利号:US-9893302-B2
优先权日:2013-03-06
标 题:Heterocyclic fluorescent dyes and method of production thereof
发明人：GRYKO DANIEL T; GRZYBOWSKI MAREK
权利人:BASF SE
摘要:The invention relates to novel compounds of formula (III) that can be used as heterocyclic dyes of unique structure and properties. These compounds can be obtained in a three-step synthesis from simple substrates. The compounds according to the invention have excellent solubility in organic solvents and excellent film-forming properties. In addition, high efficiency of energy conversion, excellent field-effect mobility, good on/off current ratios and/or excellent stability can be observed, when the compounds according to the invention are used in organic field effect transistors, organic photovoltaics (solar cells) and photodiodes.

专利号:US-8940895-B2
优先权日:2011-12-21
标 题:Heterocyclic fluorescent dyes and method of production thereof
发明人：GRZYBOWSKI MAREK; GRYKO DANIEL T
权利人:BASF SE
摘要:The invention relates to novel compounds of formula (III) that can be used as heterocyclic dyes of unique structure and properties. These dyes can be obtained in a three-step synthesis from simple substrates.