专利号:US-6262272-B1 优先权日:1997-11-13 标题 :Method of synthesis of pyrrole amides 发明人:RAGAN JOHN ANTHONY; MAKOWSKI TERESA WOODALL; AM ENDE DAVID JON; CLIFFORD PAMELA JANE; YOUNG GREGORY RANDALL; CONRAD ALYSON KAY; EISENBEIS SHANE ALLEN; QUALLICH GEORGE JOSEPH; ALLEN DOUGLAS JOHN MELDRUM 权利人:PFIZER 摘要:A method for preparing pyrrole-carboxyamides which selectively bind to GABAa receptors; which comprises reacting 1,3-cycloakane-diones with bromoethylacetate followed by reaction of the resulting product with an acid halide followed by reaction with an aromatic amine and finally with an amonium source at an elevated temperature.
专利号:WO-9925684-A1 优先权日:1997-11-13 标题 :Method of synthesis of pyrrole amides
专利号:EP-1030838-A1 优先权日:1997-11-13 标 题 :Method of synthesis of pyrrole amides
专利号:EP-1030838-B1 优先权日:1997-11-13 标 题:Method of synthesis of pyrrole amides
专利号:RU-2194701-C2 优先权日:1995-12-18 标 题 :Derivatives of quinazoline, methods of their synthesis, pharmaceutical composition comprising thereof and method of achievement of anti-angiogenic effect and/or effect of decrease of vascular penetration with their using
参考文献:10.1055/s-2008-1077880 摘要:Muller T, Bräse S, Pierrat P, Réthoré C. Design and Efficient Synthesis of Fullerene Bismalonates as Building Blocks for Metal Organic Frameworks and Organic Nanostructures. Synlett. 2008 Jun 11;2008(11):1706–10. doi: 10.1055/s-2008-1077880.