CAS: 4931-47-9; N-(5-Methylpyridin-2-yl)Acetamide

相似化合物

5231-96-9 851914-61-9 149141-11-7

上下游产品

CAS号65478-62-8 N-(5-甲基-1-氧化物-2... | CAS号1603-41-4 2-氨基-5-甲基吡啶 | CAS号108-24-7 乙酸酐 | CAS号108-99-6 3-甲基吡啶 | CAS号75-05-8 乙腈 | CAS号3167-49-5 6-氨基烟酸 | CAS号36052-24-1 6-氨基烟酸甲酯 | CAS号329-89-5 6-氨基烟酰胺 | CAS号20173-49-3 2-氯-5-甲基吡啶-N-氧化物 | CAS号98953-23-2 6-乙酰氨基烟酸甲酯 | CAS号21550-48-1 6-乙酰氨基烟酸 | CAS号77837-05-9 6-acetamidopyri... | CAS号65478-62-8 N-(5-甲基-1-氧化物-2... | CAS号66362-95-6 5-甲基-2-氨基吡啶1-氧化物

N-(1-Hydroxy-5-Methylpyridin-2-Ylidene)Acetamide置于[pd(Dippf)Cl2],三乙胺体系中,用 乙腈 作为反应溶剂,化学反应 1.0H,以95%的收率获得产物2-乙酰氨基-5-甲基吡啶
参考文献:通过钯催化的三烷基胺转移氧化对吡啶 N-氧化物进行脱氧
标题:通过钯催化的三烷基胺转移氧化对吡啶 N-氧化物进行脱氧
摘要:描述了一种方便的化学选择性方法,用于通过转移氧化由 [pd(Oac) 2]/dppf 催化的三乙胺转移氧化吡啶 N-氧化物衍生物.
DOI:10.1055/s-0028-1083508

专利信息

专利号:US-RE42890-E
优先权日:2003-05-23
标题 :Furazanobenzimidazoles
发明人：EBERLE MARTIN; BACHMANN FELIX; STREBEL ALESSANDRO; ROY SUBHO; SRIVASTAVA SUDHIR; SAHA GOUTAM
权利人:BASILEA PHARMACEUTICA AG
摘要:The invention relates to compounds of formula (I) wherein R represents aryl or heteroaryl, X is oxygen, a carbonyl group, an oxime derivative of a carbonyl group or an α,β-unsaturated carbonyl group, and the substituents R 1 to R 6 have the meanings given in the specification, for use as medicaments, to novel compounds of formula (I), to methods of synthesis of such compounds, to pharmaceutical compositions containing compounds of formula (I), to the use of a compounds of formula (I) for the preparation of a pharmaceutical composition for the treatment of neoplastic and autoimmune diseases, and to methods of treatment of neoplastic and autoimmune diseases using such compounds of formula (I) or of pharmaceutical compositions containing same