专利号:US-6264962-B1 优先权日:1997-12-19 标 题:Use of cinnamic acid or of at least one of its derivatives in a cosmetic composition 发明人:BRETON LIONEL; GIRERD FLORENCE; RENAULT BEATRICE 权利人:OREAL 摘要:The invention relates to the use of cinnamic acid, or of at least one of its derivatives, in a cosmetic composition as an agent for promoting the synthesis of the skin's total lipids. n The invention also relates to a cosmetic composition comprising an effective amount of cinnamic acid or of at least one of its derivatives.
专利号:US-6133452-A 优先权日:1997-08-22 标题 :Synthesis of bisindolylmalimides 发明人:FAUL MARGARET MARY; WINNEROSKI JR LEONARD LARRY 权利人:LILLY CO ELI 摘要:The present invention provides for the reaction of optionally substituted indole-3-acetamides with optionally substituted methyl indole-3-glyoxyl reagent to prepare potent PKC inhibitors. The reaction is very efficient and robust macrocyclization methodology.
专利号:US-6037475-A 优先权日:1996-03-20 标题:Synthesis of indolymaleimides 发明人:FAUL MARGARET M; JIROUSEK MICHAEL R; MCDONALD III JOHN H; NEEL DAVID ANDREW 权利人:LILLY CO ELI 摘要:The present invention provides a method for synthesizing indolylmaleimides by reacting an activated maleimide preferably with an optionally substituted organometalic-3-indole in the presence of a transition metal catalyst.
专利号:US-6660283-B2 优先权日:1997-12-19 标 题 :Use of cinnamic acid, or of at least one of its derivatives in a cosmetic composition 发明人:BRETON LIONEL; GIRERD FLORENCE; RENAULT BEATRICE 权利人:OREAL 摘要:The invention relates to the use of cinnamic acid, or of at least one of its derivatives, in a cosmetic composition as an agent for promoting the synthesis of the skin's total lipids.The invention also relates to a cosmetic composition comprising an effective amount of cinnamic acid or of at least one of its derivatives.
专利号:US-5859261-A 优先权日:1997-03-20 标 题 :Synthesis of indolylmaleimides 发明人:FAUL MARGARET M; JIROUSEK MICHAEL R; MCDONALD III JOHN H; NEEL DAVID ANDREW 权利人:LILLY CO ELI 摘要:The present invention provides a method for synthesizing indolylmaleimides by reacting an activated maleimide preferably with an optionally substituted organometallic-3-indole in the presence of a transition metal catalyst.
专利号:US-5990319-A 优先权日:1996-08-23 标 题 :Synthesis of bisindolylmaleimides 发明人:FAUL MARGARET MARY; WINNEROSKI JR LEONARD LARRY 权利人:LILLY CO ELI 摘要:The present invention provides for the reaction of optionally substituted indole-3-acetamides with optionally substituted methyl indole-3-glyoxyl reagent to prepare potent PKC inhibitors. The reaction is a very efficient and robust macrocyclization methodology.
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合成参考文献
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