109-01-3 + 97746-91-3 = 82419-36-1 反应条件:1.1 Reagents: Triethylamine Solvents: Dimethyl Sulfoxide1.2 Solvents: Methanol,Water 标题:Synthesis Of Fluoroquinolone Antimicrobial Agent Ofloxacin 作者:Wang,Erhua; Et Al 参考文献:Zhongguo Yiyao Gongye Zazhi 日期:1991 卷标:22(9) 页码:385-7]
109-01-3 + 86760-99-8 = 82419-36-1 反应条件:1.1 Solvents: Acetonitrile1.2 Reagents: Hydrochloric Acid Solvents: Water 标题:An Efficient Synthesis Of Ofloxacin And Levofloxacin From 3,4-Difluoroaniline 作者:Adrio,Javier; Et Al 参考文献:Heterocycles 日期:1999 卷标:51(7) 页码:1563-1572]
= 82419-36-1 反应条件:1.1 Reagents: Sodium Hydride Solvents: 1,4-Dioxane1.2 Reagents: Sodium Hydroxide Solvents: Water 标题:Pyridonecarboxylic Acids As Antibacterial Agents. Part 6. A New Synthesis Of 7H-Pyrido[1,2,3-De][1,4]Benzoxazine Derivatives Including An Antibacterial Agent,Ofloxacin 作者:Egawa,Hiroshi; Et Al 参考文献:Chemical & Pharmaceutical Bulletin 日期:1986 卷标:34(10) 页码:4098-102]
= 82419-36-1 反应条件:1.1 Solvents: Dimethyl Sulfoxide1.2 Reagents: Sodium Hydroxide Solvents: Dimethyl Sulfoxide,Water 标题:Trimethylsilyl Esters And Solvates Of Chelates Of Quinoline-3-Carboxylic Acids,And Their Preparation And Use In A Process For Quinolone Antibacterials. 参考文献:Spain]
专利号:US-5521310-A 优先权日:1992-10-07 标 题 :Process to obtain benzoxazines to be used for the synthesis of ofloxazine, levofloxazine and derivatives 发明人:CARRETERO GONZALVEZ JUAN-CARLO; VICIOSO SANCHEZ MERCEDES; GARCIA RUANO JOSE-LUIS 权利人:ETILO DERIVADOS 摘要:A process to obtain benzoxazines useful for the synthesis of Ofloxazine, Levofloxazine and derivatives. The benzoxacines (I) where Xb is an halogen and R 1 is H, alkyl or alkenyl of up to 6 atoms of C or aryl, can be obtained by means of cycling a compound of formula (II) through the reaction with triphenylphosphine and ethyl azodicarboxilate. The compounds of formula (II) can be obtained through the reaction of a compound (III) with an adequate epoxide. Through the use of the adequate chiral epoxide it is possible to obtain the enantiomerically desired intermediate and, therefore and selectively, it is possible to obtain the desired final product with the adequate enantiomeric form without the need to carry out a resolution stage. n The Compounds (I) are useful and key intermediates for the synthesis of the antimicrobials Oflixazine and Levofloxazine. ##STR1##
专利号:US-10925977-B2 优先权日:2006-10-05 标 题 :Efficient synthesis of chelators for nuclear imaging and radiotherapy: compositions and applications 发明人:YANG DAVID J; YU DONGFANG; THOMPSON ANDREW S 权利人:YANG DAVID J; YU DONGFANG; THOMPSON ANDREW S; CEIL POINT LLC; UNIV TEXAS 摘要:Novel methods of synthesis of chelator-targeting ligand conjugates, compositions comprising such conjugates, and therapeutic and diagnostic applications of such conjugates are disclosed. The compositions include chelator-targeting ligand conjugates optionally chelated to one or more metal ions. Methods of synthesizing these compositions in high purity are also presented. Also disclosed are methods of imaging, treating and diagnosing disease in a subject using these novel compositions, such as methods of imaging a tumor within a subject and methods of diagnosing myocardial ischemia.
专利号:US-2024197774-A1 优先权日:2021-04-16 标 题:Synthesis of Antimicrobial PVP-coated Bismuth Nanoparticles 发明人:LOPEZ-RIBOT JOSE; VAZQUEZ-MUNOZ ROBERTO 权利人:UNIV TEXAS 摘要:Described herein is a facile, fast, and economical method for the synthesis of BAL-mediated PVP-BiNPs, using basic laboratory instruments and reagents readily available in most laboratories.
专利号:US-2011087037-A1 优先权日:2007-10-31 标题:Synthesis of ring b abeo-sterols as novel inhibitors of mycobacterium tuberculosis 发明人:RODRIGUEZ-PIERLUISSI ABIMAEL D; WEI XIAOMEI 权利人:INTELLECTUAL PROPERTY AND TECHNOLOGY VIC OFF OF 摘要:Novel 3β-hydroxy-Δ 5 -steroid analogs possessing a contracted cyclopentane B-ring provide good inhibitory activity against Mycobacterium tuberculosis . The 5(6→7)abeo-sterol nucleus present in compounds of the invention represents a novel scaffold for the development of new antitubercular agents.
专利号:US-10308663-B2 优先权日:2015-06-16 标题:Inhibitors of PTP4A3 for the treatment of cancer 发明人:LAZO JOHN S; SHARLOW ELIZABETH R; MCQUEENEY KELLEY E; WIPF PETER; SALAMOUN JOSEPH M 权利人:LAZO JOHN S; SHARLOW ELIZABETH R; MCQUEENEY KELLEY E; WIPF PETER; SALAMOUN JOSEPH M; UNIV VIRGINIA PATENT FOUNDATION; UNIV OF PITTSBURGH —OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 摘要:The invention provides protein tyrosine phosphatase inhibitor compounds, Their pharmaceutical compositions, uses, and methods of use, such as in the treatment of various cancers, and process for making the compounds. Also disclosed is an improved synthesis of protein tyrosine phosphatase inhibitor and precursor compound thienopyridone (5).
专利号:US-9982005-B2 优先权日:2013-04-04 标 题 :Macrolides and methods of their preparation and use 发明人:MYERS ANDREW G; SEIPLE IAN BASS; ZHANG ZIYANG 权利人:HARVARD COLLEGE 摘要:Provided herein are methods of preparing macrolides by the coupling of an eastern and western half, followed by macrocyclization, to provide macrolides, including both known and novel macrolides. Intermediates in the synthesis of macrolides including the eastern and western halves are also provided. Pharmaceutical compositions and methods of treating infectious diseases and inflammatory conditions using the inventive macrolides are also provided. A general diastereoselective aldol methodology used in the synthesis of the western half is further provided.
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合成参考文献
摘要:S10 | SWISSPHARMA | Pharmaceutical List with Consumption Data | DOI:10.5281/zenodo.2623484