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参考文献: Oxazolidinone Derivatives As Antimicrobials[fr] Derives D'Oxazolidinone Utilises Comme Agents Antimicrobiens
标题: Oxazolidinone Derivatives As Antimicrobials[fr] Derives D'Oxazolidinone Utilises Comme Agents Antimicrobiens
摘要:本发明涉及某些取代苯基噁唑烷酮以及其合成方法.本发明还涉及含有本发明化合物作为抗微生物药物的药物组合物.这些化合物是有用的抗微生物剂,对多种人类和兽医病原体有效,包括革兰氏阳性厌氧细菌,例如多重耐药葡萄球菌,链球菌和肠球菌,以及厌氧生物,例如bacterioides属和clostridia属物种,以及耐酸生物,例如结核分枝杆菌,埃维分枝杆菌和分枝杆菌属.

专利信息

专利号:US-2010286211-A1
优先权日:2004-10-08
标题:Oxazolidinone derivatives as antimicrobials
发明人：DAS BISWAJIT; AHMED SHAHADAL; YADAV AJAY SINGH; GHOSH SOMA; GUJRATI ARTI; SHARMA PANKAJ; RATTAN ASHOK
权利人:DAS BISWAJIT; AHMED SHAHADAL; YADAV AJAY SINGH; GHOSH SOMA; GUJRATI ARTI; SHARMA PANKAJ; RATTAN ASHOK
摘要:The present invention relates to certain substituted phenyl oxazolidinones and to processes for the synthesis of the same. This invention also relates to pharmaceutical compositions containing the compounds of the present invention as antimicrobials. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria, for example, multiple-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms, for example, Bacterioides spp. and Clostridia spp. species, and acid fast organisms, for example, Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.