CAS: 799247-52-2; Methyl 2-Chloro-5-(1-(((6-Methylpyridin-2-yl)Methoxy)Imino)Ethyl)Benzylcarbamate

该化合物是一种苯丙基氨基甲酸酯杀菌剂,具有广泛的抗真菌病原体活动,特别是控制灰色霉菌(Botrytis cinerea)和水果,蔬菜和装饰品等作物中的其他叶子病,其行动方式包括干扰真菌电子运输链中的复杂三型,从而阻止线虫体呼吸,提供独特的生化目标,从而提供有效保护. Pyribencarb 展出跨拉米纳运动,加强其保护和治疗效果.它因其应用率低,抗药性管理潜力和与综合虫害管理(IPM)方案的兼容性而受到重视.该化合物展示了有利的环境和毒理学特征,使它成为可持续农业的实用选择.

结构式图片

物理性质

MSDS等安全信息

欧盟法规

C&L通报

合成工艺路线路线简述

  • 1122-71-0 + 325155-30-4 = 799247-52-2
    反应条件:1.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt1.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491]

    325155-92-8 = 799247-52-2
    反应条件:1.1 Reagents: Triethylamine,Hydroxyamine Hydrochloride Solvents: Ethanol; 5 H,Rt -> Reflux2.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt2.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491]

    89-97-4 = 799247-52-2
    反应条件:1.1 30 Min; 3 H,Rt1.2 Reagents: Water; 30 Min,Rt2.1 Reagents: Aluminum Chloride Solvents: Dichloromethane; Rt2.2 Rt; 1 H,Rt; 15 H,Reflux; Reflux -> Rt2.3 Reagents: Water3.1 Reagents: Hydrochloric Acid Solvents: Water; 6 H,Rt -> Reflux4.1 Reagents: Triethylamine Solvents: Dichloromethane; 30 Min,Rt4.2 1 H,Rt; 5 H,Rt5.1 Reagents: Triethylamine,Hydroxyamine Hydrochloride Solvents: Ethanol; 5 H,Rt -> Reflux6.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt6.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491]

    714915-76-1 = 799247-52-2
    反应条件:1.1 Reagents: Triethylamine Solvents: Dichloromethane; 30 Min,Rt1.2 1 H,Rt; 5 H,Rt2.1 Reagents: Triethylamine,Hydroxyamine Hydrochloride Solvents: Ethanol; 5 H,Rt -> Reflux3.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt3.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491]

    = 799247-52-2
    反应条件:1.1 Reagents: Hydrochloric Acid Solvents: Water; 6 H,Rt -> Reflux2.1 Reagents: Triethylamine Solvents: Dichloromethane; 30 Min,Rt2.2 1 H,Rt; 5 H,Rt3.1 Reagents: Triethylamine,Hydroxyamine Hydrochloride Solvents: Ethanol; 5 H,Rt -> Reflux4.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt4.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491]

    57058-32-9 = 799247-52-2
    反应条件:1.1 Reagents: Aluminum Chloride Solvents: Dichloromethane; Rt1.2 Rt; 1 H,Rt; 15 H,Reflux; Reflux -> Rt1.3 Reagents: Water2.1 Reagents: Hydrochloric Acid Solvents: Water; 6 H,Rt -> Reflux3.1 Reagents: Triethylamine Solvents: Dichloromethane; 30 Min,Rt3.2 1 H,Rt; 5 H,Rt4.1 Reagents: Triethylamine,Hydroxyamine Hydrochloride Solvents: Ethanol; 5 H,Rt -> Reflux5.1 Reagents: Thionyl Chloride Solvents: Dichloromethane; Rt; Overnight,Rt5.2 Reagents: Potassium Carbonate Solvents: Dimethylformamide; 4 H,Rt -> 80 °C
    标题:Synthesis Of Pyribencarb And Its Bioactivity
    作者:Chai,Baoshan; Et Al
    参考文献:Nongyao 日期:2011 卷标:50(7) 页码:489-491

海关参考信息

专利信息


专利号:WO-2025056767-A1
优先权日:2023-09-15
标题 :Process for the preparation of enantiomerically enriched aliphatic amines
发明人：BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS
权利人:SYNGENTA CROP PROTECTION AG
摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.

专利号:US-9968097-B2
优先权日:2012-05-30
标题:Composition comprising a biological control agent and a fungicide selected from inhibitors of the lipid membrane synthesis, the melanine biosynthesis, the nucleic acid synthesis or the signal transduction
发明人：WACHENDORFF-NEUMANN ULRIKE; ANDERSCH WOLFRAM; STENZEL KLAUS; SPRINGER BERND
权利人:BAYER CROPSCIENCE AG
摘要:The present invention relates to a composition comprising at least one biological control agent. Furthermore, the present invention relates to the use of this composition as well as a method for reducing overall damage of plants and plant parts.

专利号:WO-2021074309-A1
优先权日:2019-10-16
标 题:1-(3-quinolyl)-3,4-dihydroisoquinoline derivatives as fungicides for combating specific phytopathogens
发明人：WEISS MATTHIAS; QUARANTA LAURA; BOU HAMDAN FARHAN; MAHAJAN ATUL; WILLIAMS SIMON; KILARU JAGADEESH; SEN INDIRA; BIERI STEPHANE; DIGGELMANN MARTIN
权利人:SYNGENTA CROP PROTECTION AG
摘要:1-(3-quinolyl)-3,4-dihydroisoquinoline derivatives of formula (I) as well as a method of combating, preventing or controlling the phytopathogens Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale), which comprises applying to the phytopathogen, to the locus of the phytopathogen, or to a plant susceptible to attack by the phytopathogen, or to propagation material thereof, a fungicidally effective amount of a 1-(3-quinolyl)-3,4-dihydroisoquinoline derivative of formula (I). The present description discloses the synthesis of exemplary compounds, formulation examples, relevant biological data (antifungal activity against Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale) when spayed on plants), as well as comparative data against three prior art compounds (e.g. pages 52 to 85; formulation examples; examples A1 to A3; table E; compounds E.01 to E.187; biological examples). Exemplary compounds are e.g.: 5-bromo-1-(8-fluoro-3-quinolyl)spiro[4H-isoquinoline-3,1'- cyclopropane] (example A1) 5-bromo-1-(8-fluoro-3-quinolyl)-3,3-dimethyl-4H-isoquinoline (example A2) 1-(8-fluoro-3-quinolyl)-3,3-dimethyl-4H-isoquinoline-5-carbonitrile (example A3)

专利号:WO-2021074311-A1
优先权日:2019-10-16
标题:1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives as fungicides for combating specific phytopathogens
发明人：WEISS MATTHIAS; QUARANTA LAURA; BOU HAMDAN FARHAN; MAHAJAN ATUL; WILLIAMS SIMON; KILARU JAGADEESH; BIERI STEPHANE; DIGGELMANN MARTIN
权利人:SYNGENTA CROP PROTECTION AG
摘要:1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives of formula (I) as well as a method of combating, preventing or controlling the phytopathogens Mycosphaerella graminicola (Septoria tritici), Fusarium culmorum, Gibberella zeae (Fusarium graminearum) and Monographella nivalis (Microdochium nivale), which comprises applying to the phytopathogen, to the locus of the phytopathogen, or to a plant susceptible to attack by the phytopathogen, or to propagation material thereof, a fungicidally effective amount of a 1-(3-quinolyl)-1,2,3,4-tetrahydroisoquinoline derivatives of formula (I). The present description discloses the synthesis of exemplary compounds, formulation examples, relevant biological data (antifungal activity against Mycosphaerella graminicola, Monographella nivalis, Fusarium culmorum and/or Gibberella zeae when spayed on plants) (e.g. pages 47 to 55; examples A1 and A2; compounds E.01 to E.17; table E). An exemplary compounds is e.g.: 3-(5-bromo-3,3-dimethyl-2,4-dihydro-1 H-isoquinolin-1-yl)-8-fluoro- quinoline (example A1)

专利号:US-2011230343-A1
优先权日:2008-10-24
标题 :Method for the Manufacture of Microparticles Comprising an Effect Substance
发明人：SCHROERS MICHAEL; DYLLICK-BRENZINGER RAINER; MERK MICHAEL; BARG HEIKO
权利人:BASF SE
摘要:A subject matter of the present invention is a process for the preparation of effect compound-comprising microparticles M comprising A) the formation of a crude suspension of microparticles A by means of enzymatic polyester synthesis in an inverse miniemulsion comprising enzyme, effect compound and polyester monomers; and B) the polymerization of wall monomers from the group consisting of ethylenically unsaturated monomers, polyisocyanates and polyepoxides in the crude suspension of microparticles A. Furthermore, the present invention relates to microparticles M which can be obtained by means of the process according to the invention and also to an agrochemical formulation comprising microparticles M. In addition, the present invention relates to the use of microparticles M prepared according to the invention as component in colorants, cosmetics, drugs, biocides, plant protection agents, fertilizers, additives for food or animal fodder, or auxiliaries for polymers, paper, textiles, leather, detergents or cleaners. Finally, the invention also relates to a method for combating undesirable plant growth, to a method for combating undesirable insect or acarid infestation on plants and/or for combating phytopathogenic fungi, and to seeds treated with the agrochemical formulation.

专利号:US-9706777-B2
优先权日:2012-05-30
标题:Composition comprising a biological control agent and a fungicide selected from inhibitors of amino acid or protein biosynthesis, inhibitors of ATP production and inhibitors of the cell wall synthesis
发明人：WACHENDORFF-NEUMANN ULRIKE; ANDERSCH WOLFRAM; STENZEL KLAUS; SPRINGER BERND
权利人:BAYER CROPSCIENCE AG
摘要:The present invention relates to a composition comprising at least one biological control agent. Furthermore, the present invention relates to the use of this composition as well as a method for reducing overall damage of plants and plant parts.

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