专利号:US-9809566-B2 优先权日:2012-09-06 标题:Organocatalytic process for asymmetric synthesis of decanolides 发明人:RAWAT VARUN; DEY SOUMEN; SHELKE ANIL MARUTI; SURYAVANSHI GURUNATH MALLAPPA; SUDALAI ARUMUGAM 权利人:COUNCIL SCIENT IND RES 摘要:The present invention discloses organocatalytic process for asymmetric synthesis of highly enantioselective decanolide compounds in high yield with >99% ee. Further, the present invention disclose cost effective, improved organocatalytic process for asymmetric synthesis of highly enantioselective decanolides compounds from non-chiral, cheap, easily available raw materials.
专利号:US-3655715-A 优先权日:1969-07-15 标 题:Synthesis of n-substituted 2-aminoethanethiosulfuric acids 发明人:KLAYMAN DANIEL L; GILMORE W FRANKLIN 权利人:US ARMY 摘要:A PROCESS FOR THE SYNTHESIS OF N-SUBSTITUTED 2-AMINOETHANETHIOSULFURIC ACIDS OF THE FORMULA: R-NH-CH2-CH2-SSO3H WHEREIN R REPRESENTS ALKYL OR PHENYL ALKYL BY REACTING AMMONIUM THIOSULFATE WITH A 1-SUBSTITUTED AZIRIDINE. THE COMPOUNDS MADE BY THIS PROCESS ARE EFFECTIVE ANTIRADIATION AGENTS FOR ANIMALS.
专利号:US-9150498-B2 优先权日:2011-10-25 标题:Process for the preparation of oseltamivir and methyl 3-epi-shikimate 发明人:RAWAT VARUN; DEY SOUMEN; ARUMUGAM SUDALAI 权利人:COUNCIL SCIENT IND RES 摘要:The present invention discloses high yielding enantioselective process for synthesis of Oseltamivir from readily available starting material, cis-1,4-butene diol. The process features incorporation of chirality using sharpless asymmetric epoxidation (AE) and diastereoselective Barbier allylation and construction of cyclohexene carboxylic acid ester core through a ring closing metathesis (RCM) reaction. Further also disclosed herein is synthesis of (−)-methyl 3-epi-shikimate.
专利号:US-2004226330-A1 优先权日:2001-03-05 标 题:Anionic polymers composed of dicarboxylic acids and uses thereof 发明人:SANDERS JOHN LARRY; MAZO GRIGORY; MAZO JACOB 摘要:Biodegradable anionic polymers are disclosed which include recurring polymeric subunits preferably made up of dicarboxylic monomers such as maleic anhydride, itaconic anhydride or citraconic anhydride. Free radical polymerization is used in the synthesis of the polymers. The polymers may be complexed with ions and/or mixed with fertilizers or seeds to yield agriculturally useful compositions. The preferred products of the invention may be applied foliarly or to the earth adjacent growing plants in order to enhance nutrient uptake by the plants.
专利号:US-2004226331-A1 优先权日:2001-03-05 标题:Anionic polymers composed of dicarboxylic acids and uses thereof 发明人:SANDERS JOHN LARRY; MAZO GRIGORY; MAZO JACOB 摘要:Biodegradable anionic polymers are disclosed which include recurring polymeric subunits preferably made up of dicarboxylic monomers such as maleic anhydride, itaconic anhydride or citraconic anhydride. Free radical polymerization is used in the synthesis of the polymers. The polymers may be complexed with ions and/or mixed with fertilizers or seeds to yield agriculturally useful compositions. The preferred products of the invention may be applied foliarly or to the earth adjacent growing plants in order to enhance nutrient uptake by the plants.
专利号:US-2004230020-A1 优先权日:2001-03-05 标题 :Anionic polymers composed of dicarboxylic acids and uses thereof 发明人:SANDERS JOHN LARRY; MAZO GRIGORY; MAZO JACOB 摘要:Biodegradable anionic polymers are disclosed which include recurring polymeric subunits preferably made up of dicarboxylic monomers such as maleic anhydride, itaconic anhydride or citraconic anhydride. Free radical polymerization is used in the synthesis of the polymers. The polymers may be complexed with ions and/or mixed with fertilizers or seeds to yield agriculturally useful compositions. The preferred products of the invention may be applied foliarly or to the earth adjacent growing plants in order to enhance nutrient uptake by the plants.
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合成参考文献
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