专利号:US-8114993-B2 优先权日:2007-02-06 标题:Use of aryl chlorides in palladium-catalyzed C-H bond functionalization 发明人:DAUGULIS OLAFS; CHIONG HENDRICH 权利人:DAUGULIS OLAFS; CHIONG HENDRICH; UNIV HOUSTON SYSTEM 摘要:A one-step method for efficiently converting carbon-hydrogen bonds into carbon-carbon bonds using chloroarenes and palladium catalysts is disclosed. This method allows faster introduction of complex molecular entities, a process that would otherwise require many more steps. This invention is particularly relevant for the organic synthesis of complex molecules such as, but not limited to, pharmacophores.
专利号:US-11542283-B2 优先权日:2018-05-28 标题 :Synthesis of peptide borate ester compound and use thereof 发明人:QIN YANRU 权利人:JIANGSU CHIA TAI FENGHAI PHARMACEUTICAL CO LTD 摘要:Provided are a peptide borate ester compound or a pharmaceutically acceptable salt thereof, a preparation method therefor, and pharmaceutical use thereof. The peptide borate ester compound or pharmaceutically acceptable salt thereof has a structure as shown in Formula (I), and is useful in the preparation of proteasome inhibitors to treat solid tumors and hematoma.
专利号:US-2021214377-A1 优先权日:2018-05-28 标题 :Synthesis of peptide borate ester compound and use thereof
专利号:CN-119320374-A 优先权日:2024-11-04 标 题 :A method for photocatalytic synthesis of 3-sulfonyl-substituted chromone derivatives
专利号:WO-2019228299-A1 优先权日:2018-05-28 标 题:Synthesis and uses of peptide borate ester compound
专利号:CN-115215798-B 优先权日:2022-06-10 标题 :A kind of aromatic cyanide synthesis method of inert olefins
参考标题:Palladium Catalyzed Regioselective C4‐arylation And Olefination Of Indoles And Azaindoles 作者:Neetipalli Thrimurtulu,Arnab Dey,Anurag Singh,Kuntal Pal,Debabrata Maiti,Chandra M. R. Volla |发布日期:2019.3.15 摘要:A Convergent Strategy For The Synthesis Of Biologically Relevant C4‐substituted Indole Scaffolds Was Demonstrated Using Pd(II)‐catalyzed Remote C−h Functionalization Of Indoles And Azaindoles. The Reaction Displays High Regioselectivity For The C4‐position Of Indole‐3‐carbaldehydes Using Glycine As An Inexpensive Transient Directing Group. Notable Features Of This Transformation Include The Selective
合成参考文献
摘要:Sumida, Y.; Ohmiya, H., Science of Synthesis Knowledge Updates, (2022) 3, 43. 摘要:Weibel, J.-M.; Blanc, A.; Pale, P., Science of Synthesis Knowledge Updates, (2018) 1, 90. 摘要:Mérour, J.-Y.; Joseph, B., Science of Synthesis Knowledge Updates, (2016) 3, 113. 摘要:Zhdankin, V. V., Science of Synthesis Knowledge Updates, (2015) 1, 240. 摘要:Zhdankin, V. V., Science of Synthesis Knowledge Updates, (2015) 1, 234.