CAS: 35216-39-8; 3-(Methylsulfonyl)Aniline

上下游产品

CAS号2976-32-1 1-甲砜基-3-硝基苯 | CAS号1783-81-9 3-氨基茴香硫醚 | CAS号3937-95-9 3-Nitrophenylsu... | CAS号33951-33-6 2-甲砜基溴苯 | CAS号19614-16-5 2-溴茴香硫醚 | CAS号5335-40-0 3-甲砜基苯磺酰氯 | CAS号2976-32-1 1-甲砜基-3-硝基苯 | CAS号771573-22-9 3-(甲基磺酰基)苯甲胺 | CAS号125802-65-5 9-benzyl-2-chlo... | CAS号22821-75-6 3-(甲基磺酰基)苯甲腈

苯甲砜置于ferrous(II) Sulfate Heptahydrate,Hydroxylamine Triflate体系中,化学反应 2.0H,以77%的收率获得产物3-甲砜基苯胺
参考文献:六氟异丙醇中的芳族ch-h胺化†
标题:六氟异丙醇中的芳族ch-h胺化†
摘要:我们报道了一种直接自由基芳族胺化反应,与现有技术相比,该反应提供了未保护的苯胺,并且底物范围得到了改善.溶剂六氟异丙醇与阳离子物种的阴离子之间的氢键可增加反应性,并可以合理地增加底物范围.我们的发现可能与一般直接c-h功能化的芳烃的自由基添加有关.
DOI:10.1039/c8Sc04966A

专利信息

专利号:US-7700654-B2
优先权日:2005-02-05
标 题:Isolation of N-butylbenzenesulfonamide, synthesis of benzenesulfonamide derivatives, and use of N-butylbenzenesulfonamide and benzenesulfonamide derivatives for treating benign prostatic hyperplasia and/or prostate carcinoma
发明人：HOFFMANN HANS-RAINER; MATUSCH RUDOLF; BANIAHMAD ARIA
权利人:LOHMANN THERAPIE SYST LTS
摘要:A process for isolating N-butylbenzenesulfonamide (NBBS) from biological material, the chemical synthesis of benzenesulfonamide derivatives, the use of NBBS and benzenesulfonamide derivatives for treating benign prostatic hyperplasia and/or prostate carcinoma, the production of medicaments for the treatment thereof, and the use of NBBS and benzenesulfonamide derivatives as a lead substance in the development of active substances for treating benign prostatic hyperplasia and/or prostate carcinoma are provided.

专利号:US-2008177107-A1
优先权日:2005-02-05
标题 :Isolation of N-Butylbenzenesulfonamide, Synthesis of Benzenesulfonamide Derivatives, and Use of N-Butylbenzenesulfonamide and Benzenesulfonamide Derivatives for Treating Benign Prostatic Hyperplasia and/or Prostate Carcinoma

专利号:CA-2596618-A1
优先权日:2005-02-05
标题:Isolation of n-butylbenzenesulfonamide, synthesis of benzenesulfonamide derivatives, and use of n-butylbenzenesulfonamide and benzenesulfonamide derivatives for treating benign prostatic hyperplasia and/or prostate carcinoma

专利号:US-6417195-B1
优先权日:1999-02-22
标题 :Isoquinoline derivatives and isoquinoline combinatorial libraries
发明人：LEBL MICHAL
权利人:LION BIOSCIENCE AG
摘要:The present invention provides the synthesis of heterocyclic compounds based on the isoquinoline ring. More specifically, the invention provides novel isoquinoline derivatives as well as novel libraries comprised of such compounds.

专利号:CA-2596618-C
优先权日:2005-02-05
标 题:Isolation of n-butylbenzenesulfonamide, synthesis of benzenesulfonamide derivatives, and use of n-butylbenzenesulfonamide and benzenesulfonamide derivatives for treating benign prostatic hyperplasia and/or prostate carcinoma

专利号:US-5874443-A
优先权日:1995-10-19
标 题:Isoquinoline derivatives and isoquinoline combinatorial libraries
发明人：KIELY JOHN S; GRIFFITH MICHAEL C
权利人:TREGA BIOSCIENCES INC
摘要:The present invention provides the synthesis of heterocyclic compounds based on the isoquinoline ring. More specifically, the invention provides novel isoquinolines as well as novel libraries comprised of many such compounds, and methods of synthesizing the libraries.