CAS: 1621862-70-1; Cpi-1205

专利信息

专利号:US-10457640-B2
优先权日:2016-10-19
标 题:Synthesis of inhibitors of EZH2
发明人：VASWANI RISHI G; HEWITT MICHAEL CHARLES
权利人:CONSTELLATION PHARMACEUTICALS INC
摘要:Provided herein are synthetic methods for the preparation of EZH2 inhibitors.

专利号:US-2019233375-A1
优先权日:2016-10-19
标题:Synthesis of inhibitors of ezh2

专利号:US-2025236590-A1
优先权日:2021-10-20
标题 :A method for the preparation of indole-3-carboxylic acid derivatives
发明人：DEB INDUBHUSAN
权利人:DEB INDUBHUSAN
摘要:The present invention provides a new synthetic method for the preparation of building block indole-3-carboxylic acid (ICA) derivatives used as a key starting material to produce several artificial drugs. An efficient, safe, operationally simple, cost-effective method for the preparation of several ICA derivatives has been introduced in a very simple way. Utilizing easily available starting material, reagent, and solvent several key starting materials of ICA derivatives have been synthesized rapidly indicates the novel method is functional group tolerable. The preparation process does not involve use of any reducing agents or transition metals in the economically viable and operationally simple condition in one pot. ICA derivatives have been generated from isatin derivative in one step and this methodology is important with a wide range of applications from the drug development and material synthesis CN point of view.

专利号:EP-3529242-A1
优先权日:2016-10-19
标 题 :Synthesis of inhibitors of ezh2

专利号:WO-2018075598-A1
优先权日:2016-10-19
标题 :Synthesis of inhibitors of ezh2