CAS: 1837-57-6; 7-Ethoxyacridine-3,9-Diamine 2-Hydroxypropanoate

乳酸,依沙吖啶 以 水,异丙醇 用作溶剂,以12.58 G的收率获得乳酸依沙吖啶
参考文献:Cn115850171
标题:Cn115850171

专利信息

专利号:US-2022395555-A1
优先权日:2020-06-11
标题:Derivatives of antibiotics
发明人：FARBER BORIS; FARBER SOF'YA; MARTYNOV ARTUR VIKTOROVICH
权利人:FARBER BORIS; FARBER SOFYA; MARTYNOV ARTUR VIKTOROVICH
摘要:Field of application: The invention relates to chemistry, pharmacy and cosmetology, allows to synthesize of supramolecular structure on base antibiotics derivatives for use in pharmacy, cosmetology and pharmacy. n The essence of the invention: a new derivatives of antibiotics based on supramolecular structures and a method for their preparation, characterized in that the supramolecular structures are obtained by combinatorial synthesis of an antibiotic from one source molecule with two or more groups available in the reaction for covalent modification, at least with two different modifiers simultaneously, this creates a mixture of modified derivatives of the original molecule, with a maximum variety of derivatives with forming new supramolecular structure, and as biologically active substances to create pharmaceutical compositions use such supramolecular structure without separation into individual components, and in the reaction a combinatorial mixture of modified derivatives of the original molecule is formed antibiotic, the maximum number of combinations. n Technical result: modified combinatorial derivatives of antibiotics with antimicrobial and antifungal activity against multiresistant and pan drug resistance strains of microorganisms and fungi. Means have a wide spectrum of action, and the supramolecular and combinatorial structure of their tens and hundreds of derivatives eliminates the resistance of microorganisms.

专利号:US-9987208-B2
优先权日:2013-04-04
标题 :Elastin synthesis/regeneration promoting agent
发明人：NISHIZAKI TOMOYUKI; TANAKA AKITO
权利人:NISHIZAKI BIOINFORMATION RES INSTITUTE
摘要:8-[2-(2-Pentyl-cyclopropylmethyl)-cyclopropyl]-octanoic acid (DCP-LA) has an action to promote synthesis and regeneration of elastin, and is useful as an agent for the prophylaxis or improvement of wrinkles, and an anti-aging drug.

专利号:US-4129648-A
优先权日:1977-11-21
标 题 :Method for reducing endogenous prostaglandin synthesis
发明人：COLLIER HARRY O J; SAEED SHEIKH A; SCHNEIDER CYRIL; MANNUZZA FRANK
权利人:COLLIER HARRY O J; SAEED SHEIKH A; SCHNEIDER CYRIL; MANNUZZA FRANK
摘要:A high molecular weight extract of mammalian blood plasma and serum proteins of the group Cohn fraction IV, Cohn subfraction IV1, IV4 and haptoglobin, have been found to contain activity which inhibits endogenous prostaglandin synthetase. This extract is therefore of utility in treating or alleviating pathological conditions associated with excessive or unbalanced snythesis of endogenous prostaglandins, for example, in reducing bronchoconstriction or treating arthritis. For this purpose, the extract may be administered by injection, by inhalation, or topically.

专利号:US-3763009-A
优先权日:1970-10-05
标 题 :Synthesis process for the production of ascorbic acid glucoside
发明人：SUZUKI Y; MIYAKE T
权利人:HAYASHIBARA CO
摘要:The present invention relates to a process for the improvement of the oxidation resistance of ascorbic acid by subjecting a mixture of ascorbic acid, maltose and/or oligosaccharides to the action of an enzyme derived from genera Asperigillus, Penicillium or others to convert the mixture enzymatically into ascorbic acid glucoside.

专利号:CN-106458847-B
优先权日:2014-05-29
标 题:Synthesis of Novel Diamine and Liquid Crystal Aligning Agent Using It

专利号:RU-2039742-C1
优先权日:1992-09-14
标 题:Method of synthesis of 2-ethoxy-6-nitro-9-aminoacridine