专利号:US-9597327-B2 优先权日:2005-05-25 标 题:Synthesis of (R)-N-methylnaltrexone 发明人:DOSHAN HAROLD D; PEREZ JULIO 权利人:PROGENICS PHARM INC 摘要:This invention relates to stereoselective synthesis of R-MNTX and intermediates thereof, pharmaceutical preparations comprising R-MNTX or intermediates thereof and methods for their use.
专利号:US-2010055750-A1 优先权日:2008-09-03 标 题:Polyester synthesis 发明人:WOSNICK JORDAN H 权利人:XEROX CORP 摘要:The present disclosure provides for enzymatic polymerization to produce polyester resins suitable for use in manufacturing toners. In embodiments, crystalline copolymers, which are polyesters, may be synthesized from lactones, cyclic anhydrides, cyclic carbonates, and combinations thereof. These crystalline copolymers, in turn, may be utilized in the synthesis of toner particles.
专利号:US-9174904-B1 优先权日:2014-07-15 标 题 :Synthesis of 2,2-bis(3-phenyl-4-hydroxyphenyl) propane (PHP) 发明人:CHANDRA GIRISH; SAIT MEERAKANI MOHAMED ALI; TANWAR AKHILESH; SHETTY SHARANKUMAR 权利人:SABIC GLOBAL TECHNOLOGIES BV 摘要:Disclosed herein are ortho aryl substituted bisphenol monomers that exhibit a lower binding energy to estradiol related receptors. The monomers are provided by the condensation of a ketone and phenol in the presence of an acid catalyst.
专利号:US-7825268-B2 优先权日:2003-12-23 标 题:Alkoxylactones, alkoxylactams and alkoxythiolactams for controlling processes based on microbial interaction 发明人:STUMPE STEFAN; BREVES ROLAND; HUCHEL URSULA; JANSSEN FRANK; HAETZELT ANDRE 权利人:HENKEL AG & CO KGAA 摘要:Compounds of the Formula I, n nwherein A 1 is O or NH; A 2 is O or S; each of R 1 and R 2 is independently hydrogen, a methyl or C 2 -C 8 -saturated or mono- or doubly unsaturated, branched or linear hydrocarbon group; and R 3 is a C 1 -C 18 -saturated or mono- or doubly unsaturated, branched or linear hydrocarbon group wherein, each of R 1 , R 2 and R 3 comprises a heteroatom selected from the group consisting of O and S in the chain and/or is mono- or multiply-substituted by a substituent selected from the group consisting of halogen, hydroxy, C 1 -C 6 -alkyl, trifluoromethyl, C 1 -C 6 -alkoxy, C 6 -C 10 -aryl, and C 1 -C 6 -alkyl-C 6 -C 10 -aryl are useful for controlling the interaction process between microorganisms such as in the development and/or maturation of biofilms; multicellular swarm behavior; the concerted development of antibiotic resistances; the concerted synthesis of antibiotics; the concerted synthesis of pigments; the concerted production of extracellular enzymes; or the concerted production of virulence factors.
专利号:WO-2024246279-A1 优先权日:2023-05-31 标 题 :Lightening compositions and use of compounds as depigmenting agents 发明人:HUYSSEUNE SANDRA; VEITHEN ALEX 权利人:CHEMCOM SA 摘要:The present invention relates to a lightening composition comprising a lightening effective amount of a compound of formula (I), or a tautomer, a stereoisomer, a hydrate, a solvate, a salt, or a polymorph thereof, wherein R1, R2, R3, R4, R5, R6, R7, m and n are as defined in the description and claims. The present invention also relates to a compound of formula (I2) or a tautomer, a stereoisomer, a hydrate, a solvate, a salt, or a polymorph thereof, wherein R1, R2, R3, R4, R5, R6, and R7 are as defined in the description and claims. The present invention also relates to the use of at least one compound of formula (I) or any subgroup thereof, or mixtures thereof, as depigmenting agent. The present invention also relates to the use of at least one compound of formula (I) or any subgroup thereof, or the use of the lightening composition, for preventing and/or reducing pigmentation of normal skin. The present invention also relates to the use of at least one compound, or the use of the lightening composition according to the first aspect, for decreasing the amount of melanin in melanocytes, for decreasing melanin synthesis, for impairing melanin transport and/or for impairing the distribution of melanin in suprabasal layers.
专利号:US-7674904-B2 优先权日:2005-05-25 标 题 :Synthesis of R-N-methylnaltrexone
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合成参考文献
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