CAS: 1177865-17-6; N6-(2-((5-(Diethylamino)Pentan-2-yl)Amino)-6-Methylpyrimidin-4-yl)-2-Methylquinoline-4,6-Diamine Trihydrochloride

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    主要参考文献


    1: Zhang Y, Zhang H, Zhao S, Qi Z, He Y, Zhang X, Wu W, Yan K, Hu L, Sun S, Tang X, Zhou Q, Chen F, Gu A, Wang L, Zhang Z, Yu B, Wang D, Han Y, Xie L, Ji Y. S-Nitrosylation of Septin2 Exacerbates Aortic Aneurysm and Dissection by Coupling the TIAM1-RAC1 Axis in Macrophages. Circulation. 2024 Jun 11;149(24):1903-1920. doi: 10.1161/CIRCULATIONAHA.123.066404. Epub 2024 Feb 15. 44(9):1263-1271. doi: 10.1248/bpb.b21-00054. Epub 2021 Jun 23. 15(1):40931. doi: 10.1038/s41598-025-24830-x.
    4: Levay M, Krobert KA, Wittig K, Voigt N, Bermudez M, Wolber G, Dobrev D, Levy FO, Wieland T. NSC23766, a widely used inhibitor of Rac1 activation, additionally acts as a competitive antagonist at muscarinic acetylcholine receptors. J Pharmacol Exp Ther. 2013 Oct;347(1):69-79. doi: 10.1124/jpet.113.207266. Epub 2013 Jul 25. 24(6):3582-3592. doi: 10.1111/jcmm.15049. Epub 2020 Feb 10.
    6: Hou H, Chávez AE, Wang CC, Yang H, Gu H, Siddoway BA, Hall BJ, Castillo PE, Xia H. The Rac1 inhibitor NSC23766 suppresses CREB signaling by targeting NMDA receptor function. J Neurosci. 2014 Oct 15;34(42):14006-12. doi: 10.1523/JNEUROSCI.1659-14.2014.

    合成参考文献


    参考文献:10.1189/jlb.0108064
    摘要:Sundararaj KP, Samuvel DJ, Li Y, Nareika A, Slate EH, Sanders JJ, Lopes-Virella MF, Huang Y. Simvastatin suppresses LPS-induced MMP-1 expression in U937 mononuclear cells by inhibiting protein isoprenylation-mediated ERK activation. J Leukoc Biol. 2008 Oct;84(4):1120–9.
    参考文献:10.1186/s13567-018-0551-9
    摘要:Szczepanski A, Owczarek K, Milewska A, Baster Z, Rajfur Z, Mitchell JA, Pyrc K. Canine respiratory coronavirus employs caveolin-1-mediated pathway for internalization to HRT-18G cells. Veterinary Research. 2018 Jul 03;49(1):55. doi: 10.1186/s13567-018-0551-9.
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