专利号:WO-9636627-A1 优先权日:1995-05-19 标 题 :Collection of activated glycoside compounds and their biological use 发明人:ANDERSON MARK BRIAN; MUSSER JOHN H 权利人:GLYCOMED INC 摘要:The present invention relates to the field of combinatorial carbohydrate chemistry and involves the modification of organic molecules and/or the synthesis of large numbers of products comprising carbohydrate and/or glycominetic entities. More specifically, the present invention relates to activated carbon glycosides useful for the modification of organic molecules by incorporation of carbohydrate units, providing the synthesis of large numbers of products having novel chemical characteristics. The present invention further relates to methods for the generation of chemical compounds comprising carbon glycosides. Methods are disclosed to provide large arrays of molecules and to identify species that act as agonists or antagonists of various biological, chemical, and other activities.
专利号:US-9777034-B2 优先权日:2013-05-21 标题 :Modular synthesis of amphiphilic Janus glycodendrimers and their self-assembly into glycodendrimersomes 发明人:PERCEC VIRGIL 权利人:UNIV PENNSYLVANIA 摘要:The invention concerns compounds of the formula (I) wherein: Y 1 and Y 2 are independently a monosaccharide or disaccharide; X 1 and X 2 are independently —(R 9 —O) m —, —(R 10 ) p —, —O—(R 11 —O) q —, —R 16 —O—R 17 —O— or a covalent bond; Q 1 and Q 2 are independently a nitrogen-containing heterocycle moiety; Z 1 and Z 2 are independently —(O—R 7 )—, —(O—C(â•?O)—R 8 )a-, —O—C(â•?O)—R 12 —C(=0)-R 13 —, —O—C(â•?O)—R 14 —C(â•?O)—R 15 or a covalent bond; R 7 -R 17 are each independently C 1 -C 6 alkyl; R 1 -R 6 are each independently a linear or branched alkyl group; b, c, d, e, f, and g are 0 or 1, provided b+c+d equals at least 2 and e+f+g equals at least 2; and a, m, p, and q are each an integer from 1-6.
专利号:RU-2165266-C1 优先权日:2000-06-28 标题 :Method of synthesis of [2-18f]-2-deoxyglucose
专利号:US-2016108076-A1 优先权日:2013-05-21 标题:Modular synthesis of amphiphilic janus glycodendrimers and their self-assembly into glycodendrimersomes
专利号:WO-2014190024-A1 优先权日:2013-05-21 标题 :Modular synthesis of amphiphilic janus glycodendrimers and their self-assembly into glycodendrimersomes
参考标题:A Concise Synthesis Of Oligosaccharides Derived From Lipoarabinomannan (Lam) With Glycosyl Donors Having A Nonparticipating Group At C2 作者:Zhihao Li,Changping Zheng,Marco Terreni,Teodora Bavaro,Matthieu Sollogoub,Yongmin Zhang |发布日期:2020.4.16 摘要:Is One Of The Top Ten Leading Causes Of Death Over The World, And Lipoarabinomannan (Lam) Has Been Confirmed To Play Significant Roles In This Process. In This Study, A Convenient Synthetic Approach Has Been Developed For The Synthesis Of Oligosaccharides Derived From Lam Starting With Commercially Available Substrates And Reagents. The Key Steps For Stereoselective Construction Of Glycosidic Bonds By
合成参考文献
摘要:Kryczka, B.; Lewkowski, J.; Zawisza, A., Science of Synthesis, (2007) 29, 992. 摘要:Kryczka, B.; Lewkowski, J.; Zawisza, A., Science of Synthesis, (2007) 29, 997. 摘要:Robina, I.; Vogel, P., Science of Synthesis, (2008) 37, 755.