CAS: 217500-96-4; Tulathromycin A

上下游产品

propylamine carbonic acid benzyl ester 4-dimethylamino-2-[2-ethyl-3,4,10-trihydroxy-13-(8-methoxy-4,8-dimethyl-1,5-dioxa-spiro[2.5]°Ct-6-yloxy)-3,5,8,10,12,14-hexamethyl-15-oxo-1-oxa-6-aza-cyclopentadec-11-yloxy]-6-methyl-tetrahydro-pyran-3-yl ester erythromycin A 9-(E)-oxime 9-Deoxo-9a-aza-9a-homoerythromycin A

阿奇霉素 A置于palladium 10% On Activated Carbon,Potassium Tert-Butylate,氢气,Potassium Carbonate,戴斯-马丁氧化剂,Sodium Sulfate体系中,用 四氢呋喃,二氯甲烷,水,二甲基亚砜,异丙醇,丙酮 用作溶剂,-85.0~65.0 °C,250.0 Kpa 条件下,反应 4.5H,反应生成托拉菌素 A
参考文献:泰拉菌素中间体的盐
标题:泰拉菌素中间体的盐
摘要:本发明公开了一种制备泰拉菌素的中间体的盐,具体来说该盐为草酸盐,及其制备方法和在制备泰拉菌素的方法中的应用.

专利信息

专利号:WO-2025056767-A1
优先权日:2023-09-15
标题 :Process for the preparation of enantiomerically enriched aliphatic amines
发明人：BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS
权利人:SYNGENTA CROP PROTECTION AG
摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.

专利号:CN-119638694-A
优先权日:2018-11-16
标 题 :Improved synthesis of key intermediates for KRAS G12C inhibitor compounds

专利号:CN-114728960-B
优先权日:2019-11-14
标 题:Improved synthesis of KRAS G12C inhibitor compounds

专利号:CN-113015724-B
优先权日:2018-11-16
标题 :Improved synthesis of key intermediates for KRAS G12C inhibitor compounds

专利号:CN-119638693-A
优先权日:2018-11-16
标 题 :Improved synthesis of key intermediates for KRAS G12C inhibitor compounds

专利号:CN-104119413-B
优先权日:2014-07-29
标题:A kind of synthesis method of tulamycin residue marker