专利号:WO-2025056767-A1 优先权日:2023-09-15 标题 :Process for the preparation of enantiomerically enriched aliphatic amines 发明人:BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS 权利人:SYNGENTA CROP PROTECTION AG 摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.
专利号:WO-2011067757-A1 优先权日:2009-12-06 标题 :INSECTICIDAL COMPOSITIONS OF CHITIN SYNTHESIS INHIBITORS (CSIs) AND THE ENTOMOPATHOGENIC FUNGUS NOMURAEA RILEYI 发明人:APPLEBAUM SHALOM W; ICHELCZIK DANA; BARAZANI AVNER 权利人:MAKHTESHIM CHEM WORKS LTD; YISSUM RES DEV CO; APPLEBAUM SHALOM W; ICHELCZIK DANA; BARAZANI AVNER 摘要:The present invention discloses a pesticidal composition comprising a combination of a chitin synthesis inhibitor (CSI) and the fungus Nomuraea rileyi, wherein this composition is insecticidally effective and contains an insecticidally effective amount of a chitin synthesis inhibitor and an insecticidally effective amount of the fungus Nomuraea rileyi. Also are disclosed a method of treating or preventing pest infestation in a plant or in an environment in which this plant is grown, by contacting the plant or environment with the pesticidal composition of the invention, and a method for reducing the amount of CSI required to control insects, and the use of the pesticidal composition of the invention in controlling insects in a plant or an environment of the plant.
专利号:US-10906880-B2 优先权日:2016-01-26 标题:Kind of isothiazole oxime ether-containing strobilurin derivatives and its preparation methods and application 发明人:FAN ZHIJIN; CHEN LAI; GUO XIAOFENG; ZHU YUJIE; QIAN XIAOLIN; MA LIUYONG; ZHANG NAILOU; WANG HAIXIA; ZHANG ZHIMING; XU JINGHUA; SONG YINQI 权利人:UNIV NANKAI 摘要:The present invention is that provided a synthesis method of a series of isothiazole oxime ether containing strobilurin derivatives IV. The present invention relates to 3,4-dichloroisothiazolyl oxime ether strobilurin derivatives, and their chemical structural formula is as shown by IV. n n n n n n n n n n The invention discloses the structural formula of the above compound, the synthesis method and the use as an insecticide, a fungicide, an anti-plant virus agent, and an agriculturally acceptable auxiliary or synergist and a commercial insecticide. The use of a fungicide, an anti-plant virus agent and an acaricide in combination for controlling agricultural, forestry, horticultural plant pests, diseases, virus diseases and preparation methods.
专利号:US-7628979-B1 优先权日:2005-04-20 标题 :Use of calco oil blue V in bait formulations for marking and controlling subterranean termites 发明人:MORALES-RAMOS JUAN A; ROJAS MARIA G 权利人:US AGRICULTURE 摘要:Termite bait matrix containing cellulose, calco oil blue V (solvent blue 58 or 9,10-anthracenedione, 1,4-bis[(2-ethylhexyl)amino]), and optionally a termite toxicant (e.g., chitin synthesis inhibitor). Methods of monitoring termite activity in a region involving placing a termite bait matrix in the region and assessing the presence of termites at the site of the termite matrix, the termite bait matrix contains cellulose and 9,10-anthracenedione, 1,4-bis[(2-ethylhexyl)amino]. Methods of killing termites, involving placing a termite bait matrix in a termite habitat and allowing termites to feed on the bait matrix, the termite bait matrix contains cellulose, 9,10-anthracenedione, 1,4-bis[(2-ethylhexyl)amino], and a termite toxicant (e.g., chitin synthesis inhibitor).
专利号:WO-02087337-A3 优先权日:2001-05-01 标 题:Pesticidal compositions comprising a chitin synthesis inhibitor and piperonyl butoxide 发明人:VERBRUGGEN LUC ROSALIA MICHAEL 权利人:JANSSEN PHARMACEUTICA NV; VERBRUGGEN LUC ROSALIA MICHAEL 摘要:The present invention relates to pesticide compositions and particularly to compositions which are able to provide an improved protecting effect against invertebrates such as insects and acari. More particularly, the present invention relates to synergistic pesticide compositions comprising a chitin synthesis inhibitor and piperonyl butoxide for protecting any living or non-living material, such as crops, plants, fruits, seeds, building parts made of wood, thatch or the like, biodegradable material and textiles against deterioration due to the action of pests such as insects and for treating animals, especially mammals, gallinaceae and anatidae, against such harmful invertebrates. This invention thus relates to the field of protection of plants, crops, warm-blooded animals, food, building materials and textiles through the control of pests. The chitin biosynthesis inhibitors are specifically, bistrifluron, buprofezin, chlorfluazuron, diflubenzuron, flucycloxuron, flufenoxuron, hexaflumuron, lufenuron, novaluron, teflubenzuron or triflumuron. Preferred is flufenoxuron.
专利号:US-2007232495-A1 优先权日:2006-03-24 标题:Compositions and methods to add value to plant products, increasing the commercial quality, resistance to external factors and polyphenol content thereof 发明人:NAPPA ALVARO O; LORENZINI FELIPE C; SANHUEZA ANDRES L 权利人:NAPPA ALVARO O; LORENZINI FELIPE C; SANHUEZA ANDRES L 摘要:The invention is related to compositions and methods that naturally protect plant tissues against ultraviolet radiation and temperature, thus giving protection against sunburn to plants, plant parts, fruits and/or flowers during their development. The invention is also related to compositions and methods to naturally improve the color of plants, plant parts, fruits and/or flowers by inducing the natural synthesis of flavonoids and anthocyanins present in plants. Likewise, the present invention is directed to improving the nutritional value of plants, plant parts, fruits and/or flowers by increasing the normal levels of polyphenolic compounds, especially flavonoids, present therein. Additionally, the present invention is related to compositions and methods that give more resistance to plants, plant parts, fruits and/or flowers against pathogens as bacteria and fungi. Finally, the present invention is related to plants, plant parts, fruits, flowers and/or propagating material treated with the compositions described in the present document.
1: Rouabhi R, Berrebbah H, Djebar MR. Evaluation of toxicity of two pesticides: flucycloxuron and diflubenzuron on a cellular model, Paramecium sp. Commun Agric Appl Biol Sci. 2006;71(2 Pt A):83-90. doi: 10.1021/jf304468b. Epub 2013 Jan 10. doi: 10.1021/jf200395g. Epub 2011 Mar 25. doi: 10.1021/jf801901h. doi: 10.1007/s00216-011-5699-3. Epub 2012 Jan 20.
合成参考文献
参考文献:10.1007/s10493-005-1423-3 摘要:Pree DJ, Whitty KJ, Van Driel L. Baseline Susceptibility and Cross Resistances of Some New Acaricides in the European Red Mite, Panonychus ulmi*. Experimental and Applied Acarology. 2005 Dec;37(3-4):165. doi: 10.1007/s10493-005-1423-3.