欧盟法规
ECHA物质C&L通报上下游产品
2-pyrrole aldehyde 2,4,5-triiodo-3-formylpyrrole (+)-D-glucosamine hydr°Chloride -α-D-glucopyranose2-deoxy-2-(3'-oxo-1'-propen-1'-yl)amino-α-D-glucopyranosepyrrole3-formyl-1-(4-methylphenyl)sulfonylpyrrole tert-butyl 3-formylpyrrole-1-carboxylate (Z)-3-(1H-Pyrrol-3-yl)-acrylic acid methyl ester (R)-5-acetamidomethyl-3-(3-fluoro-4-(3-formylpyrrol-1-yl)phenyl)isoxazoline 合成工艺路线路线简述
- 合成目标产物 Pyrrole-3-Carboxaldehyde 主要起始原料 4-Formyl-1H-Pyrrole-2-Carboxylic Acid
- (文献来源)合成步骤主要原料 4-Formyl-1H-Pyrrole-2-Carboxylic Acid
专利信息
专利号:US-7339065-B2
优先权日:2003-07-21
标题 :Design and synthesis of optimized ligands for PPAR
发明人:AVERY MITCHELL A; PERSHADSINGH HARRIHAR A
权利人:BETHESDA PHARMACEUTICALS INC; UNIV MISSISSIPPI
摘要:This invention provides new chemical entities useful for treating a variety of clinical disorders including those that are influenced by the activity of peroxisome proliferator activated receptors (PPAR). The structures of the compounds and methods to design, make and use the compounds are provided. Compounds and methods for administering therapeutic compositions comprising the compounds in cases of the disease psoriasis are provided. An exemplary compound having the formula compound is 5adamantan-2-yl-pentanoic acid {2-[4-(2,4-dioxo-thiazolidin-5-yl-methyl)-phenoxy]-ethyl}-methyl-amide is provided.
专利号:US-2010286211-A1
优先权日:2004-10-08
标题:Oxazolidinone derivatives as antimicrobials
发明人:DAS BISWAJIT; AHMED SHAHADAL; YADAV AJAY SINGH; GHOSH SOMA; GUJRATI ARTI; SHARMA PANKAJ; RATTAN ASHOK
权利人:DAS BISWAJIT; AHMED SHAHADAL; YADAV AJAY SINGH; GHOSH SOMA; GUJRATI ARTI; SHARMA PANKAJ; RATTAN ASHOK
摘要:The present invention relates to certain substituted phenyl oxazolidinones and to processes for the synthesis of the same. This invention also relates to pharmaceutical compositions containing the compounds of the present invention as antimicrobials. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria, for example, multiple-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms, for example, Bacterioides spp. and Clostridia spp. species, and acid fast organisms, for example, Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.
专利号:US-2007099969-A1
优先权日:2003-07-21
标题 :Design and synthesis of optimized ligands for ppar
专利号:CN-114539240-B
优先权日:2022-01-05
标 题:Synthesis of 3D non-fullerene receptor small molecule and application of 3D non-fullerene receptor small molecule in ternary organic solar cell
专利号:US-6852711-B2
优先权日:1998-09-11
标题:HIV protease inhibitors
发明人:BOYER JR FREDERICK EARL; DOMAGALA JOHN MICHAEL; ELLSWORTH EDMUND LEE; GAJDA CHRISTOPHER ANDREW; HAGEN SUSAN ELIZABETH; LOVDAHL MICHAEL JAMES; LUNNEY ELIZABETH ANN; MARKOSKI LARRY JAMES; PRASAD JOSYULA VENKATA NAGENDR; TAIT BRADLEY DEAN
权利人:AGOURON PHARMA
摘要:The present invention relates to novel dihydropyrones with tethered heterocycles having improved pharmacologic properties which potently inhibit the HIV aspartyl protease blocking HIV infectivity. The dihydropyrones are useful in the development of therapies for the treatment of viral infections and diseases, including AIDS. The present invention is also directed to methods of synthesis of the dihydropyrones and intermediates useful in the preparation of the final compounds.
专利号:CN-105646453-A
优先权日:2015-12-25
标题 :Synthesis of 5-(2-fluorophenyl)-N-methyl-1-(3-pyridylsulfonyl)-1H-pyrrole-3-methylamine fumarate TAK438