CAS: 17061-62-0; Bis(4-Methoxybenzyl)Amine

相似化合物

854391-95-0 14429-02-8 197728-27-1

上下游产品

CAS号3261-60-7 N-(4-甲氧基亚苄基)-4-甲氧基苄胺 | CAS号123-11-5 4-甲氧基苯甲醛; 对甲氧基苯... | CAS号2393-23-9 对甲氧基苄胺 | CAS号3717-21-3 Benzaldehyde,4-... | CAS号109163-43-1 4-methoxy-N-(4-... | CAS号2746-25-0 4-甲氧基溴苄 | CAS号2038-57-5 3-苯基丙基胺 | CAS号874-90-8 4-甲氧基苯甲腈 | CAS号3424-93-9 4-甲氧基苯甲酰胺

4-甲氧基苄胺置于甲醇,Sodium Tetrahydroborate,Sodium Sulfate体系中,用 二氯甲烷 用作溶剂,化学反应生成双-(4-甲氧基苄基)-胺
参考文献:[2]轮烷内葡糖酰胺的反应性:高反应性α-酮酰胺的机械键控制化学选择性合成及其光触发环化
标题:[2]轮烷内葡糖酰胺的反应性:高反应性α-酮酰胺的机械键控制化学选择性合成及其光触发环化
摘要:葡糖酰胺的机械联锁对于它们化学选择性氧化为 β,γ-不饱和 α-酮酰胺至关重要.这些前所未有的物种令人满意地用于蓝光驱动的环化中,通过 Norrish/yang Ii 型反应的两种模式以不同方式提供羟基-2-氮杂环丁酮或恶唑烷酮.这种行为与相同反应条件下非互锁底物的行为截然不同.
Doi:10.1002/anie.202302681

专利信息

专利号:US-9926291-B2
优先权日:2007-03-27
标 题 :Synthesis of thiohydantoins
发明人：OUERFELLI OUATHEK; DILHAS ANNA; YANG GUANGBIN; ZHAO HONG
权利人:SLOAN KETTERING INST CANCER RES
摘要:A novel synthesis of the anti-androgen, A52, which has been found to be useful in the treatment of prostate cancer, is provided. A52 as well as structurally related analogs may be prepared via the inventive route. This new synthetic scheme may be used to prepare kilogram scale quantities of pure A52.

专利号:US-12172982-B2
优先权日:2020-08-12
标 题:Synthesis of quinazoline compounds
发明人：LIM NGIAP-KIE; SHEN JEFF; SIROIS LAUREN ELIZABETH; TIMMERMAN JACOB C; TRACHSEL ETIENNE; WHITE NICHOLAS ANDREW; XU JIE; ZHANG HAIMING; BACHMANN STEPHAN; BIGLER RAPHAEL; CLAGG KYLE BRADLEY PASCUAL; DIPASQUALE ANTONIO GIOVANNI; GOSSELIN FRANCIS; ORCEL UGO JONATHAN; MEIER ROLAND CHRISTOPH
权利人:GENENTECH INC; HOFFMANN LA ROCHE
摘要:Provided herein are methods of synthesizing quinazoline compounds comprising at least one atropisomeric center.

专利号:US-2025101021-A1
优先权日:2022-06-14
标 题:Methods of making tolebrutinib
发明人：BAILLY FRÉDÉRIC; BENELLI CHRISTOPHE; BORIE CYRIL; BOSCH MICHAËL; CABOS CLAUDE; CHARAUDEAU ALEXIS; JANSSENS LAURENCE; PACQUET FRANÇOIS; RODIER FABIEN; SALLÉ LAURENT; SODO ALFRED; VIGNE SYLVIE
权利人:PRINCIPIA BIOPHARMA INC
摘要:Disclosed herein are improved synthetic routes for making (R)-1-(1-acryloylpiperidin-3-yl)-4-amino-3-(4-phenoxyphenyl)-1 H-imidazo[4,5-c]pyridin-2(3H)-one (tolebrutinbib). Also disclosed herein are novel compounds used in the synthesis of of (R)-1-(1-acryloylpiperidin-3-yl)-4-amino-3-(4-phenoxyphenyl)-1 H-imidazo[4,5-c]pyridin-2(3H)-one.

专利号:US-12071422-B2
优先权日:2022-02-07
标 题 :Process for synthesis of quinazoline compounds
发明人：LEBL RENE; LIM NGIAP KIE; MEIER ROLAND CHRISTOPH; ORCEL UGO JONATHAN; SEDELMEIER JOERG; SHEN JEFF; SIROIS LAUREN ELIZABETH; TIMMERMAN JACOB C; TRACHSEL ETIENNE; WHITE NICHOLAS ANDREW; XU JIE; ZHANG HAIMING; BACHMANN STEPHAN; BASS THOMAS MICHAEL; BIGLER RAPHAEL; BURKHARD JOHANNES ADRIAN; CLAGG KYLE BRADLEY PASCUAL; GOSSELIN FRANCIS; HAN CHONG; KALDRE DAINIS; KELLY SEAN M; HEROLD SEBASTIAN; LEITNER CHRISTIAN
权利人:GENENTECH INC; HOFFMANN LA ROCHE
摘要:Provided herein are methods to synthesize compounds useful in the treatment of cancer where such compounds comprise a quinazolinyl core moiety and at least one stereoisomeric or atropisomeric moiety.

专利号:WO-2008119015-A2
优先权日:2007-03-27
标 题 :Synthesis of thiohydantoins

专利号:US-8987452-B2
优先权日:2007-03-27
标 题:Synthesis of thiohydantoins