📜4-(2-Acetylamino-Phenylsulfanyl)-N,N-Dimethyl-3-Nitro-Benzenesulfonamide置于sodium Hydroxide体系中,用 乙醇,丙酮 作为反应溶剂,化学反应生成 硫丙拉嗪 参考文献:Synthesis And Comparison Of Activity Of 2-And 3-Dimethylsulfamidophenothiazine Derivatives 标题:Synthesis And Comparison Of Activity Of 2-And 3-Dimethylsulfamidophenothiazine Derivatives 摘要: DOI:10.1007/bf00771334
专利号:US-2008214827-A1 优先权日:2004-02-03 标 题:Synthesis of Cyanoimino-Benzoimidazoles 发明人:GOEHRING R RICHARD; WHITEHEAD JOHN; SHAO BIN 权利人:EURO CELTIQUE SA 摘要:Disclosed in certain embodiments is a process for synthesizing a compound of formula (V) and salts thereof.
专利号:US-7300639-B2 优先权日:2002-12-03 标 题:Process for removing metals from liquids 发明人:LIU WANSHENG 权利人:BRISTOL MYERS SQUIBB CO 摘要:A process is provided for removing one or more metals from liquids. Also provided is a process for the synthesis of aP2 inhibiting compounds having the formula (I) n nwherein R 1 , R 2 , R 3 , R 4 , HET, and X-Z are as described herein, which process comprising the step of removing one or more metals from a solution of the compound of formula I or an intermediate or precursor thereof. The processes for removing metal comprise the step of contacting the liquid with a solid extractant comprising a metal-binding functionality.
专利号:EP-3103803-B1 优先权日:2008-10-27 标 题 :Intermediates for the synthesis of mtor kinase inhibitors
专利号:CA-2555219-A1 优先权日:2004-02-03 标 题 :Synthesis of cyanoimino-benzoimidazoles
专利号:US-11759496-B2 优先权日:2016-05-10 标题:Compounds and pharmaceutical use thereof in the treatment of cancer 发明人:SUSIN SANTOS A; KAROYAN PHILIPPE; MERLE-BERAL HÉLÈNE 权利人:KAROYAN PHILIPPE 摘要:The present invention relates to a compound or a pharmaceutical salt thereof comprising a hexapeptide sequence of formula (I), its method of synthesis and its use in anticancer therapy. The invention also relates to a pharmaceutical composition for use in the treatment of cancer comprising at least one soluble peptide according to the invention or at least one acid nucleic according to the invention or at least one expression vector according to the invention, or at least one host cell according to the invention and a pharmaceutically acceptable carrier.
专利号:US-2023271983-A1 优先权日:2020-07-29 标题 :Functionalized isonitriles and products, preparation and uses thereof 发明人:SOTELO PÉREZ EDDY; AZUAJE GUERRERO JHONNY ALBERTO; MAJELLARO MARIA 权利人:UNIV SANTIAGO COMPOSTELA 摘要:The present invention relates to functionalized isonitrile compounds, formed by means of multicomponent environmentally friendly reactions, suitable for coupling to functional molecules such as biomolecules, APIs, chromophore and fluorophore molecules. The invention also relates to conjugates between said isonitrile compounds and functional molecules, which are useful in the synthesis of pharmaceutic drugs or tools, fluorescent molecules and labels, polymeric smart materials. The invention furthermore provides a kit for the in-vitro preparation of the functionalized isontrile compounds and conjugates. The invention also contemplates the medical use of said compounds and conjugates.
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合成参考文献
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