专利号:US-2025223262-A1 优先权日:2022-03-31 标 题 :Synthesis of morphinans with reduced herg activity and mop binding 发明人:LAMMERT ECKHARD; SCHOLZ OKKA; OTTER SILKE; HEREBIAN DIRAN; HOFFMANN TORSTEN; SANZ MIGUEL ANGEL; KRAMP LAURENZ; LEVY LAURA MARIANA; HRISTEVA STANIMIRA 权利人:HEINRICH HEINE UNIV DUESSELDORF; DEUTSCHE DIABETES FORSCHUNGSGESELLSCHAFT E V; TAROS CHEMICALS GMBH & CO KG 摘要:The invention relates to morphinan-derivatives, processes for their preparation, medicaments containing them and the use of these morphinan-derivatives for the preparation of medicaments.
专利号:US-12291505-B2 优先权日:2016-07-04 标题 :Methods for the synthesis of deuterated dextromethorphan 发明人:JOHNSON MATT; ZHAO CUNXIANG; MENG WEIHUA; LU ZHIJUN; LI YAN 权利人:AVANIR PHARMACEUTICALS INC 摘要:The application describes methods for making a deuterated dextromethorphan of Formula (I), deuterated dextromethorphan produced by these methods, and pharmaceutically acceptable salts thereof.
专利号:US-2024124402-A1 优先权日:2016-07-04 标 题:Methods for the synthesis of deuterated dextromethorphan
专利号:US-2024067608-A1 优先权日:2016-07-04 标 题:Methods for the synthesis of deuterated dextromethorphan
专利号:EP-3478664-B1 优先权日:2016-07-04 标题 :Methods for the synthesis of deuterated dextromethorphan
专利号:US-2019241525-A1 优先权日:2016-07-04 标题:Methods for the synthesis of deuterated dextromethorphan
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合成参考文献
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