CAS: 845870-47-5; 3-(Ethylsulfonyl)Phenylboronic Acid

该化合物是一种碳酸衍生物,在苯环上具有乙基硫基替代物,使其成为铃木-米亚乌拉交叉相交反应的宝贵中间体.用电阻燃的磺酰基组增强了反应性,促进了双亚烯化合物合成中高效的C-C债券形成.在标准条件下的稳定性以及与各种催化剂和溶剂的兼容性有助于其在制药和农用化学研究中的效用.该化合物的界定完善结构和一贯纯度确保了复杂的有机转化的可复制结果.其多功能性延伸到了物质科学的应用,成为功能化芳香系统的一个建筑块.

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CAS号1005499-49-9 Methyl 3'-(ethy...

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    专利号:US-9834551-B2
    优先权日:2013-04-18
    标 题 :Substituted pyrrolo[2,3-b]pyrazines and substituted pyrazolo[3,4-b]pyridines as ITK and JAK kinase inhibitors
    发明人：VANKAYALAPATI HARIPRASAD; YERRAMREDDY VENKATAKRISHNAREDDY; GANGIREDDY PARAMAREDDY; APPALANENI RAJENDRA P
    权利人:ARRIEN PHARMACEUTICALS LLC
    摘要:The present invention relates to compounds described by Formula I: n nsalts thereof, their synthesis, and their use as ITK and JAK3 inhibitors including such compounds and methods of using said compounds in the treatment of various diseases and or disorders such disease associated with abnormal cell growth such as autoimmune, inflammation, rheumatoid arthritis, systemic lupus erythematosus, atherosclerosis, ulcerative colitis, psoriatic arthritis, psoriasis, Crohn's, metabolic and cancer diseases. The present invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention and methods of using the compositions and processes for preparing the compounds of the invention.

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    合成参考文献


    参考文献:10.1055/s-0034-1380547
    摘要:Synthesis of an Aurora Kinase B Inhibitor. Synfacts. 2015 Apr 17;11(05):0456. doi: 10.1055/s-0034-1380547.
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