CAS: 13472-85-0; 5-Bromo-2-Methoxypyridine

相似化合物

55849-30-4 13472-60-1 870521-31-6

上下游产品

CAS号624-28-2 2,5-二溴吡啶 | CAS号124-41-4 甲醇钠 | CAS号1628-89-3 2-甲氧基吡啶 | CAS号67-56-1 甲醇 | CAS号53939-30-3 5-溴-2-氯吡啶 | CAS号13466-38-1 2-羟基-5-溴吡啶 | CAS号74-88-4 碘甲烷 | CAS号6628-77-9 5-氨基-2-甲氧基吡啶 | CAS号39856-50-3 5-溴-2-硝基吡啶 | CAS号34851-41-7 四丁基甲醇铵 溶液 | CAS号380917-97-5 吡仑帕奈 | CAS号381233-78-9 5-(2-吡啶基)-1,2-二... | CAS号902130-87-4 6-甲氧基-3-吡啶乙酸 | CAS号913836-17-6 5-溴-2-羟基异烟酸甲酯 | CAS号445264-61-9 2-甲氧基吡啶-5-硼酸频哪醇酯 | CAS号219671-80-4 4-(6-甲氧基吡啶-3-基)苯甲酸 | CAS号312300-42-8 6-甲氧基吡啶-3-磺酰氯 | CAS号81971-39-3 1-甲基-5-溴吡啶-2(1H)-酮 | CAS号6628-77-9 5-氨基-2-甲氧基吡啶 | CAS号65873-72-5 6-甲氧基-3-吡啶甲醛

2-甲氧基吡啶置于1,3-二溴-5,5-二甲基海因体系中,用80 %的收率获得5-溴-2-甲氧基吡啶
参考文献:用于区域选择性芳香族溴化的高度稳定的碳硼烷基连接金纳米催化剂
标题:用于区域选择性芳香族溴化的高度稳定的碳硼烷基连接金纳米催化剂
摘要:据公开,碳硼烷可生成高度稳定的核-卫星结构的 Cb@aunp.它们能够在恶劣条件下抑制活性物质的溶解,并实现了无偏芳烃的区域选择性溴化,其p : O选择性与最佳选择性非酶催化系统中的选择性相当(如果不是优于那些).
Doi:10.1002/anie.202409283

专利信息

专利号:US-8742118-B2
优先权日:2011-10-27
标题 :Methods for preparing intermediates of perampanel
发明人：FONTANA FRANCESCO; STABILE PAOLO
权利人:F I S —FABBRICA ITALIANA SINT S P A
摘要:Methods for the synthesis of 2-alkoxy-5-(pyridin-2-yl)pyridine of formula I n nor salts thereof are provided.

专利号:US-7884125-B2
优先权日:2008-04-30
标 题:Straightforward entry to 7-azabicyclo[2.2.1]heptane-1-carbonitriles and subsequent synthesis of epibatidine analogues
发明人：STEVENS CHRISTIAN; HEUGEBAERT THOMAS
权利人:UNIV GENT
摘要:The present invention relates to a group of substituted-7-azabicyclo-[2.2.1]heptyl derivatives with biological activity. The present invention also relates to synthetic methods for producing said substituted-7-azabicyclo-[2.2.1]heptyl derivatives. The present invention also relates to certain intermediates for producing such substituted-7-azabicyclo-[2.2.1]heptyl derivatives, as well as a synthetic method for producing such intermediates. The present invention also relates to pharmaceutical compositions comprising such substituted-7-azabicyclo-[2.2.1]heptyl derivatives, as well as their use as medicaments for the treatment of diseases mediated by a Nicotinic Acetylcholine Receptor or a receptor being a member of the Neurotransmitter-gated Ion Channel Superfamily, such as pain, Alzheimer's disease, Parkinson's disease, schizophrenia, epilepsy and nicotine addiction.

专利号:US-10111867-B2
优先权日:2015-02-17
标题:Process and intermediates for the preparation of perampanel
发明人：MAROM EHUD; RUBNOV SHAI
权利人:MAPI PHARMA LTD
摘要:The present invention describes a process for the synthesis of 3-(2-cyanophenyl)-5-(2-pyridyl)-1-phenyl-1,2-di-hydro-pyridin-2-one (Perampanel) represented by the structure of formula (1), and salts thereof, especially salts with pharmaceutically acceptable acids. The present invention further relates to certain intermediates formed and/or used in such process.

专利号:US-9695147-B2
优先权日:2013-07-25
标题 :Process for the preparation of perampanel
发明人：BUCHLOVIC MARIAN
权利人:TEVA PHARMACEUTICALS INT GMBH
摘要:The present invention provides intermediates useful for the synthesis of Perampanel and processes employing said intermediates for preparing Perampanel. The invention also provides processes for making the intermediates, crystalline forms of the intermediates and the use of the crystalline forms for preparing Perampanel.

专利号:US-9376400-B2
优先权日:2005-06-08
标 题:Process for the synthesis of triazoles
发明人：CHEN SHILI; LOU RONGLIANG; WU YUSHENG; ZHOU JIACHENG; HANSELMANN ROGER
权利人:MELINTA THERAPEUTICS INC
摘要:The present invention relates to processes for the preparation of triazoles. These compounds are useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents.

专利号:JP-2012197307-A
优先权日:2006-06-30
标 题 :Synthesis of diethyl {[5- (3-fluorophenyl) -pyridin-2-yl] methyl} phosphonate used in the synthesis of himbacine analogues