CAS: 3705-27-9; (S)-Hexahydropyrrolo[1,2-A]Pyrazine-1,4-Dione

相似化合物

19179-12-5 2873-36-1 2854-40-2

上下游产品

H-Pro-Gly-OMe (2S)-N-(N-Benzyloxycarbonylglycyl)prolinamide H-Pro-Gly-OEt N-chloroacetyl-L-proline ethyl esterN-prolylglycine (S)-2-(4-Methoxy-benzyl)-hexahydro-pyrrolo[1,2-a]pyrazine-1,4-dione (S)-°Ctahydropyrrolo[1,2-a]pyrazine cyclo(L)-Pro-(D)-Val

📜甲基1-{[(2-甲基-2-丙基)氧基]羰基}-L-脯氨酰甘氨酸酯置于三乙胺,三氟乙酸体系中,用 甲醇,二氯甲烷 用作溶剂,化学反应生成(8As)-六氢吡咯并[1,2-A]吡嗪-1,4-二酮
参考文献:由甘氨酰脯氨酸2,5-二酮哌嗪高度非对映选择性地合成环状α-氨基膦酸和α-氨基次膦酸
标题:由甘氨酰脯氨酸2,5-二酮哌嗪高度非对映选择性地合成环状α-氨基膦酸和α-氨基次膦酸
摘要:本文描述的环状α-氨基膦和α-Aminophosphinic酸的非对映选择性的第一合成(1-[r,8α小号)-3及(1-[r,8α小号)-4从甘氨酰-升-脯氨酸-2,5-二酮哌嗪(小号)-6,通过高度非对映亲核加成亚磷酸三甲酯或甲基苯基亚与手性碳正离子(的小号)-5.
Doi:10.1002/ejoc.201901439

专利信息

专利号:US-7723082-B2
优先权日:2002-06-21
标题 :Polynucleotides and polypeptides coded by said polynucleotides involved in the synthesis of diketopiperazine derivatives
发明人：GONDRY MURIEL; GENET ROGER; LAUTRU SYLVIE; PERNODET JEAN-LUC
权利人:COMMISSARIAT ENERGIE ATOMIQUE; CENTRE NAT RECH SCIENT
摘要:The invention concerns novel isolated natural or synthetic polynucleotides and polypeptides coded by said polynucleotides, involved in the synthesis of diketopiperazine derivatives, vectors comprising said polynucleotides, micro-organisms transformed with said polynucleotides, uses of said polynucleotides and said polypeptides, as well as methods for the synthesis of diketopiperazine derivatives, including cyclodipeptides and diketopiperazine derivatives 3- and 6-substituted by α,β-unsaturated amino acid side chains.

专利号:WO-2023064991-A1
优先权日:2021-10-22
标题 :Process for preparing bicyclic glycine-proline compounds and monocyclic glycine-proline intermediates thereof
发明人：SCOTT JEREMY PETER; KEEN STEPHEN PHILIP; ESPENSEN GEORGE MAX; PARRY-JONES DAVID; LAWRENCE RONNIE MAXWELL; BLOWER CLIVE JOHN
权利人:NEUREN PHARMACEUTICALS LTD
摘要:The present disclosure generally relates to a process for the synthesis of bicyclic glycine-proline compounds, and monocyclic glycine-proline intermediates thereof. In particular, the present disclosure also relates to a process for the synthesis of cyclic G-2-AllylP and its analogues. The present disclosure also relates to a process for the synthesis of optionally protected monocyclic glycine-proline intermediates. The present disclosure also relates to a process for the synthesis of esterified glycine-proline intermediates. The present disclosure also relates to compounds prepared by the processes and the use of such compounds to prepare compositions and to treat disorders.

专利号:US-2006051837-A1
优先权日:2002-06-21
标 题 :Polynucleotides and polypeptides coded by said polynucleotides involved in the synthesis of diketopiperazine derivatives

专利号:US-2007048817-A1
优先权日:2002-06-21
标 题:Polynucleotides and polypeptides coded by said polynucleotides involved in the synthesis of diketopiperazine derivatives

专利号:AU-2003255681-B2
优先权日:2002-06-21
标题:Polynucleotides and polypeptides coded by said polynucleotides involved in the synthesis of diketopiperazine derivatives

专利号:CN-103710412-A
优先权日:2013-12-11
标题 :Synthesis of salidroside catalyzed by β-glucosidase cross-linked aggregates