CAS: 1003-07-2; Isothiazol-3(2H)-One

相似化合物

25629-58-7 2682-20-4 26172-54-3

上下游产品

CAS号1668-10-6 甘氨酰胺盐酸盐 | CAS号1002-19-3 3-[(3-氨基-3-氧代丙基... | CAS号2807-36-5 Thi°Cyanic acid... | CAS号2682-21-5 2-ethyl-1,2-thi... | CAS号55512-82-8 3-溴异噻唑 | CAS号14217-66-4 3-Chloro-1,2-th... | CAS号26172-55-4 异噻唑啉酮 | CAS号42828-67-1 2-(2-chloroacet... | CAS号60666-83-3 3-(Benzyloxy)is... | CAS号61457-45-2 2-(2,2,2-trichl... | CAS号61457-46-3 2-(2-hydroxyeth...

📜甘氨酰胺盐酸盐置于磺酰氯体系中,用 Dmf (N,N-Dimethyl-Formamide) 用作溶剂,化学反应 7.5H,以90%的收率获得异噻唑-3-酮
参考文献:Imidazolo-5-Yl-2Anilino-Pyrimidines As Agents For The Inhibition Of The Cell Proliffration
标题:Imidazolo-5-Yl-2Anilino-Pyrimidines As Agents For The Inhibition Of The Cell Proliffration
摘要:该公式化合物(i):其中r1,R2,R3,R4,R5,R6,P,Q和n的定义如下,并描述了其药用盐和体内可水解酯.还描述了它们的制备过程以及它们作为药物的用途,特别是作为用于在温血动物(如人)中产生细胞周期抑制(抗细胞增殖)作用的药物.

专利信息

专利号:WO-2025085030-A1
优先权日:2023-10-18
标 题:Synthesis of semisynthetic penicillin derivatives containing hydrazone-derived thiazolidine and imidazole ring
发明人：SARIPINAR EMIN; BURAN SUMEYYE
权利人:ERCIYES UNIV
摘要:The present invention relates to the novel semi-synthetic thiazolidine and imidazole penicillin, pharmaceutically acceptable derivatives thereof and their synthesis method that may cause biologically significant changes by the N-acylation reaction of 6-aminopenicillanic (6-APA) using new trisubstituted thiazolidine and imidazole acetyl chloride derivatives. The invention also relates to pharmaceutical compositions comprising these compounds and their use for therapeutic treatment in the human or animal body.

专利号:WO-2025085026-A1
优先权日:2023-10-18
标 题:Synthesis of semisynthetic penicillin derivatives containing hydrazone-derived thiazolidine and imidazole ring
发明人：SARIPINAR EMIN; BURAN SUMEYYE
权利人:T C ERCIYES UNIV
摘要:The present invention relates to the novel semi-synthetic thiazolidine and imidazole penicillin, pharmaceutically acceptable derivatives thereof and their synthesis method that may cause biologically significant changes by the N-acylation reaction of 6-aminopenicillanic (6-APA) using new trisubstituted thiazolidine and imidazole acetyl chloride derivatives. The invention also relates to pharmaceutical compositions comprising these compounds and their use for therapeutic treatment in the human or animal body.

专利号:US-10040964-B2
优先权日:2014-02-12
标题:Use of tristyrylphenol alkoxylate sulfosuccinates in emulsion polymerization and coatings
发明人：LUEBKE GARY; RESCHAK KEITH; LUKA RENEE; KALTENBACH JARROD
权利人:STEPAN CO
摘要:Disclosed are the use of novel surfactants for the synthesis of emulsion polymer latexes, particularly those used in paints, coatings, and pressure sensitive adhesives. The surfactant compositions for emulsion polymer latexes comprise sterically bulky surfactants whose composition comprises at least one alkoxylated polyaryl substituted aromatic sulfosuccinate compound. The novel surfactants provide for the production of stable, small particle size distribution emulsion polymer latexes. The resulting latexes, when formulated into latex paint, impart improvements in water resistance as measured by film opacity, blister resistance and improved leveling characteristics, and when formulated into pressure sensitive adhesives, provide improved water resistance characteristics as measured by film opacity.

专利号:US-2009326223-A1
优先权日:2006-07-18
标题 :Synthesis of 2-amino-substituted 4-oxo-4h-chromen-8.yl-trifluoro-methanesulfonic acid esters
发明人：GRIFFIN ROGER JOHN; HARDCASTLE IAN ROBERT; DESAGE-EL MURR MARINE; RODRIGUEZ-ARISTEGUI SONSOLES; GOLDING BERNARD THOMAS
权利人:GRIFFIN ROGER JOHN; HARDCASTLE IAN ROBERT; DESAGE-EL MURR MARINE; RODRIGUEZ-ARISTEGUI SONSOLES; GOLDING BERNARD THOMAS
摘要:A method of synthesising a compound of formula (I): wherein R N1 and R N2 are independently selected from hydrogen, an optionally substituted C 1-7 alkyl group, C 3-20 heterocyclyl group, or C 5-20 aryl group, or may together form, along with the nitrogen atom to which they are attached, an optionally substituted heterocyclic ring having from 4 to 8 ring atoms; from a compound of formula (III): comprising the steps of: (a) removing the allyl group from the compound of formula (III) with appropriate reaction conditions to yield a compound of formula (II): and (b) reacting the compound of formula (II) with a triflating agent to yield a compound of formula (I).

专利号:WO-2006100479-A1
优先权日:2005-03-22
标题:Methods for the synthesis of heteroaromatic compounds
发明人：KNIGHT DAVID W
权利人:UNIV CARDIFF; KNIGHT DAVID W
摘要:Methods of making heteroaromatic compounds comprising a 5- membered ring, and dihydro forms thereof, by a metal catalysed 5-endo-cyclisation of alkynes (acetylenes) are disclosed. The methods involve the use of a catalyst comprising a silver salt, more preferably a silver (I) salt, which is employed as a heterogeneous catalyst for the cyclisation reaction. The methods can produce different types of heteroaromatic compounds and are capable of producing highly substituted products, i.e. products in which the 5-membered ring is disubstituted, trisubstituted or, with further simple reactions, tetrasubstituted. The methods described herein generally the advantages that they use conditions and reagents that are benign, cheap and flexible and amenable to scale up, and in which the only by-product is water.

专利号:US-2021386068-A1
优先权日:2018-11-07
标题 :Compositions comprising pyridine carboxylate herbicides and very long chain fatty acid (vlcfa) synthesis inhibitor herbicides
发明人：KISTER JEREMY; SATCHIVI NORBERT M
权利人:CORTEVA AGRISCIENCE LLC
摘要:Disclosed herein are compositions comprising (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof and (b) a VLCFA synthesis inhibitor herbicide. Also disclosed herein are methods of controlling undesirable vegetation, comprising applying to vegetation or an area adjacent the vegetation or applying in soil or water to control the emergence or growth of vegetation (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) a VLCFA synthesis inhibitor herbicide.