专利号:WO-2024018354-A1 优先权日:2022-07-18 标题 :A process for the synthesis of 4-alkoxy-3-hydroxypicolinic acids and intermediates thereof 发明人:MAL SANJIB; SARKAR PARANTAP; PATRA PRANAB KUMAR; KLAUSENER ALEXANDER GUENTHER MARIA 权利人:PI INDUSTRIES LTD 摘要:The present invention discloses a process for the synthesis of 4- alkoxy-3-hydroxypicolinic acids of formula (I) from 2-picolinic acid. The present invention further discloses a process for preparation of compounds of formula (iii) from compounds of formula (ii). The present invention also discloses novel intermediate compounds of formula (iii).
专利号:US-2023202980-A1 优先权日:2019-08-30 标题:N-(2-Aminophenyl)-Prop-2-Enamide Derivatives, and Uses Thereof in the Treatment of Cancer 发明人:RADHAKRISHNAN SRIDHAR; TENEN DANIEL G; LIU BEE HUI; VU LE KIM ANH; GO MEI LIN; CHAI LI; GAO CHONG; KAMAL AHMED; SUNKARI SATISH; AYINAMPUDI VENKATA SUBBARAO; SYED RIYAZ; LIU MIAO 权利人:NAT UNIV SINGAPORE; THE BRIGHAM AND WOMEN’S HOSPITAL INC; INDIAN INSTITUTE OF CHEMICAL TECH 摘要:Provided herein are N-(2-aminophenyl)-prop-2-enamide derivatives, such as those of Formula (I), methods for the synthesis thereof, and uses thereof in the treatment of cancer, such as SALL4-expressing cancer, in a cell or subject in need thereof.
专利号:US-2023018429-A1 优先权日:2019-11-22 标 题 :Process for synthesis of (3-chloro-2-pyridyl)hydrazine 发明人:CHOCKALINGAM DEVARAJAN; DUDHAT VIPUL; KHARATKAR RAJU MAHADEV; MAO JIANHUA; VEKARIYA PANKAJKUMAR; BHATT DHARMESH BALVANTRAI 权利人:FMC CORP; FMC AGRO SINGAPORE PTE LTD 摘要:Described herein are novel methods of synthesizing (3-chloro-2-pyridyl)hydrazine. Compounds prepared by the methods disclosed herein are useful for preparation of certain anthranilamide compounds that are of interest as insecticides, such as, for example, the insecticides chlorantraniliprole and cyantraniliprole.
专利号:US-3965049-A 优先权日:1972-10-24 标 题 :One-step synthesis of aromatic organic diselenides 发明人:GRUSHKIN BERNARD; SALZMAN MICHAEL N 权利人:XEROX CORP 摘要:Disclosed is a novel method for the preparation of aromatic organic diselenide compounds. The method involves reacting an alkali metal diselenide with certain halogenated aromatic compounds in dimethylformamide to form the corresponding aromatic diselenide. The use of dimethylformamide enables one to prepare certain aromatic diselenide compounds containing two replaceable halogen atoms in a one-step process.
专利号:CN-102911114-A 优先权日:2012-11-22 标题:Synthesis of 3,5-Dibromo-4-iodopyridine Catalyzed by Alkyl Silicon Reagent
专利号:CN-102898359-A 优先权日:2012-11-12 标题:Synthesis of 3,5-dibromo-4-iodopyridine
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