CAS: 19178-25-7; Pyrido[3,4-D]Pyrimidin-4(3H)-One

相似化合物

22389-85-1 171178-44-2 21038-67-5

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CAS号7579-20-6 3-氨基-4-吡啶羧酸 | CAS号64188-97-2 3-氨基异烟酸甲酯 | CAS号122-51-0 原甲酸三乙酯 | CAS号77287-34-4 甲亚胺酸 | CAS号51752-67-1 4-氯-吡啶[3,4-D]嘧啶 | CAS号88128-94-3 N-[4-(1H-imidaz...

📜3-氨基-4-吡啶羧酸 以 Formamide 用作溶剂,以72%的收率获得3,4-二氢吡啶[3,4-D]嘧啶-4-酮
参考文献:Bicyclic Compounds Capable Of Inhibiting Tyrosine Kinases Of The
标题:Bicyclic Compounds Capable Of Inhibiting Tyrosine Kinases Of The
摘要:描述了新型4-取代氨基吡啶嘧啶和4-取代氨基吡啶嘧啶抑制剂对表皮生长因子受体家族的酪氨酸激酶的作用,以及相应的药物组合物,这些药物在治疗癌症,关节炎中的滑膜侵袭,牛皮癣,血管再狭窄和血管生成方面非常有用,此外还可用于治疗胰腺炎和肾病,以及作为避孕药剂.

专利信息

专利号:US-3950160-A
优先权日:1972-09-27
标题:Inhibiting the growth of weeds with 2-substituted pyrdidopyimidines and salts thereof
发明人：ABU EL-HAJ MARWAN J; DOMINY BERYL WILLIAM
权利人:PFIZER
摘要:2-Substituted pyridopyrimidines and their alkali and alkylamine salts as herbicides, and processes for the synthesis of starting materials leading to the preparation thereof.

专利号:US-9540371-B2
优先权日:2013-04-29
标 题:Substituted quinazolin-4(3H)-ones, pyrido[3,4-d]pyrimidin-4(3H)-ones, pyrido[3,2-d]pyrimidin-4(3H)-ones and pyrido[2,3-d]pyrimidin-4(3H)-ones as positive allosteric modulators of muscarinic acetycholine receptor M1
发明人：LINDSLEY CRAIG W; CONN P JEFFREY; STAUFFER SHAUN R; PANARESE JOSEPH DAVID
权利人:UNIV VANDERBILT
摘要:In one aspect, the invention relates to 3-benzylquinazolin-4(3H)-one analogs, derivatives thereof, and related compounds, which are useful as positive allosteric modulators of the muscarinic acetylcholine receptor M 1 (mAChR M 1 ); synthesis methods for making the compounds; pharmaceutical compositions comprising the compounds; and methods of treating neurological and psychiatric disorders associated with muscarinic acetylcholine receptor dysfunction using the compounds and compositions. This abstract is intended as a scanning tool for purposes of searching in the particular art and is not intended to be limiting of the present invention. Exemplary 3-benzylquinazolin-4(3H)-one compounds include compounds of formula (I):

专利号:US-3962264-A
优先权日:1972-09-27
标 题:Process for making 2-amino nicotinonitrile
发明人：ABU EL-HAJ MARWAN J; DOMINY BERYL WILLIAM
权利人:PFIZER
摘要:2-Substituted pyridopyrimidines and their alkali and alkylamine salts as herbicides, and processes for the synthesis of starting materials leading to the preparation thereof.

专利号:US-3917624-A
优先权日:1972-09-27
标题:Process for producing 2-amino-nicotinonitrile intermediates
发明人：ABU EL-HAJ MARWAN J; DOMINY BERYL WILLIAM
权利人:PFIZER
摘要:2-Substituted pyridopyrimidines and their alkali and alkylamine salts as herbicides, and processes for the synthesis of starting materials leading to the preparation thereof.

专利号:US-3862191-A
优先权日:1972-09-27
标 题 :Pyrido{8 2,3-d{9 pyrimidin-4(3H)-one
发明人：EL-HAJ MARWAN J ABU; DOMINY BERYL WILLIAM
权利人:PFIZER
摘要:2-Substituted pyridopyrimidines and their alkali and alkylamine salts as herbicides, and processes for the synthesis of starting materials leading to the preparation thereof.

专利号:CA-2664113-C
优先权日:2006-09-22
标 题:Use of platencin and platensimycin as fatty acid synthesis inhibitors to treat obesity, diabetes and cancer