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专利号:WO-2021045879-A1 优先权日:2019-09-03 标 题 :Synthesis of deuterated aldehydes
专利号:US-2017334888-A1 优先权日:2001-07-16 标 题 :Synthesis of udp-glucose: n-acylsphingosine glucosyltransferase inhibitors
专利号:US-10000521-B2 优先权日:2013-03-15 标 题:Substituted gemcitabine bicyclic amide analogs and treatment methods using same 发明人:SUO ZUCAI; VYAVHARE VINOD P; TAGGART DAVID J 权利人:NUCORION PHARMACEUTICALS INC 摘要:In one aspect, the invention relates to substituted gemcitabine aryl amide analogs, derivatives thereof, and related compounds; synthesis methods for making the compounds; pharmaceutical compositions comprising the compounds; and methods of treating viral disorders and disorders of uncontrolled cellular proliferation using the compounds and compositions. In certain aspects, the compounds have the following structure:
专利号:CN-115368346-A 优先权日:2021-08-30 标 题 :A kind of 1,4-benzodioxane-benzimidazolium salt compound and its synthesis method and application
参考文献:10.1007/s00216-011-5225-7 摘要:Shibata S, Zhang Z, Korotkov KV, Delarosa J, Napuli A, Kelley AM, Mueller N, Ross J, Zucker FH, Buckner FS, Merritt EA, Verlinde CLMJ, Van Voorhis WC, Hol WGJ, Fan E. Screening a fragment cocktail library using ultrafiltration. Analytical and Bioanalytical Chemistry. 2011 Jul 13;401(5):1585. doi: 10.1007/s00216-011-5225-7.