Fmoc-D-葡萄糖苄基酯置于palladium On Activated Charcoal 硫酸,Ammonium Formate体系中,用 四氢呋喃,甲醇,二氯甲烷 用作溶剂,25.0 °C,199.94 Kpa 条件下,反应 6.33H,反应生成N-芴甲氧羰基-D-谷氨酸 Gamma-叔丁酯 参考文献:Synthesis Of (R)-And (S)-(Glu)Thz And The Corresponding Bisthiazole Dipeptide Of Dolastatin 3 标题:Synthesis Of (R)-And (S)-(Glu)Thz And The Corresponding Bisthiazole Dipeptide Of Dolastatin 3 摘要: Doi:10.1021/jo00374A019
专利号:US-5817751-A 优先权日:1994-06-23 标 题 :Method for synthesis of diketopiperazine and diketomorpholine derivatives 发明人:SZARDENINGS ANNA KATRIN; CAMPBELL DAVID 权利人:AFFYMAX TECH NV 摘要:The present invention relates to the areas of organic and medicinal chemistry. More specifically, the present invention is concerned with combinatorial and solid phase methods for the synthesis of diverse diketopiperazine derivatives, and the use of such methods to create libraries of diverse diketopiperazine derivatives. The present invention has application in the areas of chemical synthesis, the screening for new diketopiperazine derivatives having beneficial medical properties and the use of such screening to provide compositions and methods including diketopiperazine derivatives for treating disease.
专利号:CN-115925790-A 优先权日:2016-03-23 标 题:Method for the synthesis of α4β7 peptide antagonists
专利号:US-11879038-B2 优先权日:2019-09-09 标 题 :Supramolecular gel supported on open-cell polymer foam 发明人:JIERRY LOÃ?C; SERRA CHRISTOPHE; SCHAAF PIERRE; RODON FORES JENNIFER; BOULMEDAIS FOUZIA 权利人:UNIV STRASBOURG; CENTRE NAT RECH SCIENT; INST NAT SANTE RECH MED; CENTRE NAT RECH SCIENT; INST NAT SANTE RECH MED 摘要:The present invention relates to a polymer foam, said polymer foam comprising pores forming an open-cell polymer foam, said polymer foam comprising a supramolecular gel inside pores, and said polymer foam comprising at least one enzyme. The present invention relates to a supramolecular gel; its preparation and its applications, notably in chemical synthesis and kinetic resolution, in particular of organic compounds. The present invention also relates to flow chemistry.
专利号:CN-118085036-B 优先权日:2022-11-25 标题 :An amphiphilic D/L cyclic peptide capable of self-assembly to form a nanohelix and a synthesis and assembly method thereof