📜5-甲氧基-2-甲基-3-吲哚乙酸置于六甲基磷酰三胺,双(三甲基硅烷基)氨基钾,N,N'-二环己基碳二亚胺体系中,用 四氢呋喃 用作溶剂,化学反应生成2-[1-(4-氯苯甲酰基)-5-甲氧基-2-甲基-1H-吲哚-3-基]-1-(4-吗啉基)乙酮 参考文献:New Class Of Potent Ligands For The Human Peripheral Cannabinoid Receptor 标题:New Class Of Potent Ligands For The Human Peripheral Cannabinoid Receptor 摘要:A New Class Of Potent Ligand For The Human Peripheral Cannabinoid (Hcb(2)) Receptor Is Described. Two Indole Analogs 13 And 17 Exhibited Nanomolar Potencies (K-I) With Good Selectivity For The Hcb(2) Receptor Over The Human Central Cannabinoid (Hcb(1)) Receptor. Copyright (C) 1996 Elsevier Science Ltd Doi:10.1016/0960-894X(96)00426-X
专利号:WO-2025128903-A1 优先权日:2023-12-13 标题:Novel synthesis of substituted tricyclic compounds 发明人:WANG SILAS; BECK HILARY; RAMOS ANGEL 权利人:EIKON THERAPEUTICS INC 摘要:Processes for preparing compounds of the general formula (VIII) from a compound of general formulat (V) via the aldehyde intermediate (VI), which is combined with the compound of general formula (VII): A process for preparing the compound of formula (III) from a compound of formula (II) via the aldehyde intermediate (I), which is combined with the compound of formula (IV):
专利号:US-11891406-B2 优先权日:2019-03-14 标题:Conductivity enhancement of MOFs via development of MOFpolymer composite material 发明人:PEEDIKAKKAL ABDUL MALIK P; AL-BETAR ABDUL-RAHMAN; AL-MOUSA AMMAR HUSSAIN 权利人:UNIV KING FAHD PET & MINERALS 摘要:A method for enhancing the conductivity of MOF-5 by the development of an MOF-5 polymer composite material. The composite material incorporates a conductive polymer, preferably polyaniline, in the solvo-thermal synthesis pathway of MOF-5. The electrically conductive MOF-5 composite exhibits electric conductivity three orders of magnitude higher than that of MOF-5 while maintaining the crystallinity, robustness, and thermal stability of MOF-5.
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