欧盟法规
C&L通报专利信息
专利号:US-2023150994-A1
优先权日:2020-04-07
标 题:Methods for synthesis of chk1 inhibitors
发明人:SCHWAEBE MICHAEL; ROSNER THORSTEN; ZHAO DALIAN; MILLER ROSS; DULINA RICH; HUMORA MICHAEL; GOTTSCHLING STEPHEN E
权利人:SIERRA ONCOLOGY INC
摘要:The present technology relates to processes, compounds, compositions, and methods useful for coupling reactions. Also, the present disclosure provides for novel intermediates, compositions of matter, and processes relating to the Chk1 inhibitor, SRA737.
专利号:EP-3567040-B1
优先权日:2013-06-24
标 题 :Method for the preparation of intermediates useful for the synthesis of [1,2,4]-triazolo[4,3-a]pyridines
专利号:EP-3567040-A1
优先权日:2013-06-24
标题 :Method for the preparation of intermediates useful for the synthesis of [1,2,4]-triazolo[4,3-a]pyridines
专利号:EP-4132922-A1
优先权日:2020-04-07
标 题 :Methods for synthesis of chk1 inhibitors
专利号:WO-2025011547-A1
优先权日:2023-07-10
标 题 :Method for obtaining on-dna aromatic compound via suzuki coupling reaction and use thereof
发明人:QU YI; XIA BING; LIN SHUANG; HOU YUXIA; Zhuang Shurong; YANG MINGHUI; ZHANG HAO; GU LIANG; ZHANG PEIYU; MA JIAN
权利人:JINGTAI ZHIYAO TECH SHANGHAI CO LTD
摘要:A synthesis method for an On-DNA aromatic compound, comprising subjecting an On-DNA aromatic halide and an organic boric acid, organic borate, organic borate, borane or [Formula 1] to a coupling reaction under the catalysis of a [Pd] catalyst and an alkali, the [Pd] catalyst being a catalyst formed by 2-amino-4,6-dihydroxypyrimidine and divalent palladium. The method is simple, convenient and rapid, and can obtain On-DNA compounds via a Suzuki coupling reaction under a relatively low-temperature condition, thus rapidly expanding the range of application of DNA encoded compound libraries, and adapting to the requirements of large-batch production of DNA encoded compound libraries using multiple-well plates.
专利号:CN-116411356-A
优先权日:2021-12-29
标 题 :Synthesis method of DNA coding compound ribofuranose derivative